PASSARELLA, DANIELE
PASSARELLA, DANIELE
Dipartimento di Chimica
PROTAC-mediated degradation of peroxisomal d-aspartate oxidase: A novel strategy to modulate d-aspartate homeostasis for schizophrenia treatment
2026 M. Galli, V. Rabattoni, M. Cavinato, F. Vasile, I. Gado, K. Ulfat, H. Shehi, A. Silvani, D. Passarella, A. Citarella, L. Pollegioni, M. Nardini
Photochemical C4-Selective C-H Amination of Quinolines via N-Shift of Heteroaryl Azides
2026 A. Dimasi, A. Montoli, G. Macetti, L. Lo Presti, D. Passarella, V. Fasano
Development of In-Cell Self-Assembly Proteolysis Targeting Chimeras Exploiting the Biorthogonal Reaction Between Vinyl Boronic Acids and 1,2,4,5-Tetrazines
2026 M. Galli, L. Passarelli, E. Fassi, G. Grazioso, D. Passarella, A. Silvani
Safracin B as a Synthetic Linchpin: From Natural Product to Drug Intermediate and Beyond
2026 P. Orlando, S. Borsoi, V. Fasano, A. Citarella, P. Allegrini, D. Passarella
N‐Amidinyl‐Benzodiazaborines as Novel Boron‐Based Scaffolds: Synthesis and Application in Retromer Stabilization
2026 A. Dimasi, A. Montoli, M. Buonaguro, L. Maiorana, G. Macetti, E. Colombo, L. Muzio, G. Donati, D. Passarella, P. Seneci, V. Fasano
Rethinking Dipolar Aprotic Solvents in Medicinal Chemistry: Practical Applications of Cyrene
2026 M. Galli, A. Citarella, A. Silvani, D. Passarella
From molecular design to synthesis: novel potential degraders for Tauopathies
2026 G. Tempra, P. Bettega, E.M.A. Fassi, G. Grazioso, P. Seneci, D. Passarella
Design, synthesis and characterization of novel potential TAU-degraders
2026 G. Tempra, E.M.A. Fassi, G. Grazioso, P. Seneci, D. Passarella
Oxygen Atom Insertion Into Tetrahydroquinolines: A Skeletal Editing Approach To Unexplored 2,3-Benzoxazepines
2026 F. Migliano, A. Fiori, S. Scardigno, A. Fucina, A. Montoli, G. Macetti, L. Lo Presti, D. Passarella, V. Fasano
Stereodefined synthesis of 3-difluoromethyl-benzoxaboroles: novel antimicrobials with unlocked H-bonding
2026 A. Dimasi, A. Montoli, C. Lutti, A. Citarella, P. Ronchi, F. Castagnini, V. Mileo, G. Macetti, V. Baldelli, E. Rossi, P. Landini, D. Passarella, V. Fasano
BUILDING AND DECODING NITROGEN-CONTAINING NATURAL PRODUCTS
2026 S. Borsoi, R. Koenigs, D. Passarella
Rotational Motion in Bispidines: A Conformational Study
2025 F. Migliano, L. Pozzi, A. Citarella, G. Macetti, L. Lo Presti, D. Passarella, V. Fasano
Rotational Motion in Bispidines: A Conformational Study
2025 F. Migliano, L. Pozzi, A. Citarella, G. Macetti, L. Lo Presti, D. Passarella, V. Fasano
PROTAC technology for the degradation of hDASPO: from design to synthesis to biophysical and cellular evaluation
2025 M. Galli, A. Citarella, M. Cavinato, I. Gado, V. Rabattoni, H. Shehi, M. Nardini, A. Silvani, V. Fasano, F. Vasile, L. Pollegioni, D. Passarella
Design, synthesis and biological evaluation of PROTACs targeting hDASPO
2025 M. Galli, A. Citarella, M. Cavinato, I. Gado, V. Rabattoni, H. Shehi, M. Nardini, A. Silvani, V. Fasano, F. Vasile, L. Pollegioni, D. Passarella
Structure-Based Discovery of Hsp90/HDAC6 Dual Inhibitors Targeting Aggressive Prostate Cancer
2025 A. Citarella, S. Belluti, D. Bonanni, D. Moi, I. Piccinini, A. Rinaldi, C. Papulino, R. Benedetti, L. Cuoghi, S.D. Ciolo, A. Silvani, L. Altucci, L. Pinzi, S. Franchini, D. Passarella, C. Sorbi, C. Giannini, C. Imbriano, G. Rastelli
Revisiting the Reduction of Vinpocetine
2025 S. Borsoi, L. Pozzi, V. Fasano, A. Citarella, G. Macetti, L.L. Presti, G. Paladino, U. Ciriello, D. Passarella
An Inducible Neural Stem Progenitor Cell Model for Testing Therapeutic Interventions Against Neurodegeneration FENIB
2025 A. Giustini, A. Maiocchi, I. Serangeli, M. Pedrini, A. Quintiliani, V. Sabato, F. Bonato, P. Seneci, G. Lupo, D. Passarella, E. Miranda
Asymmetric Total Synthesis of (−)‐Glycybridin B, a Pharmacophore Screened Candidate for Tubulin Binding
2025 A. Maiocchi, M. Shevelev, Z. Boiarska, J. Estévez‐gallego, F. Bonato, P. Orlando, A. Chinosi, E. Marcone, A. Citarella, D. Horvath, M.O. Steinmetz, A.E. Prota, A. Varnek, V. Fasano, D. Passarella
Design, synthesis and in vitro validation of bivalent binders of SARS-CoV-2 spike protein: Obeticholic, betulinic and glycyrrhetinic acids as building blocks
2025 M. Pedrini, L. Pozzi, F. Sacchi, A. Citarella, V. Fasano, P. Seneci, S. Pieraccini, L. Ruberto, H. Perez Peña, A. Garzino-Demo, A. Vitiello, L. Sernicola, A. Borsetti, A. Calistri, C. Parolin, D. Passarella