PASSARELLA, DANIELE
PASSARELLA, DANIELE
Dipartimento di Chimica
Total Synthesis of an Epothilone Analogue based on the Amide‒Triazole Bioisosterism
2024 E. Colombo, D.A. Coppini, S. Borsoi, V. Fasano, R. Bucci, F. Bonato, E. Bonandi, F. Vasile, S. Pieraccini, D. Passarella
Nirmatrelvir: from discovery to modern and alternative synthetic approaches
2024 M. Galli, F. Migliano, V. Fasano, A. Silvani, D. Passarella, A. Citarella
Nicotinic Acid Derivatives As Novel Noncompetitive α-Amylase and α-Glucosidase Inhibitors for Type 2 Diabetes Treatment
2024 A. Citarella, M. Cavinato, E. Rosini, H. Shehi, F. Ballabio, C. Camilloni, V. Fasano, A. Silvani, D. Passarella, L. Pollegioni, M. Nardini
Quantitative live cell imaging of a tauopathy model enables the identification of a polypharmacological drug candidate that restores physiological microtubule interaction
2024 L. Pinzi, C. Conze, N. Bisi, G.D. Torre, A. Soliman, N. Monteiro-Abreu, N.I. Trushina, A. Krusenbaum, M.K. Dolouei, A. Hellwig, M.S. Christodoulou, D. Passarella, L. Bakota, G. Rastelli, R. Brandt
A Green Approach to Nucleophilic Aromatic Substitutions of Nicotinic Esters in Cyrene
2024 A. Citarella, M. Cavinato, A. Amenta, M. Nardini, A. Silvani, D. Passarella, V. Fasano
Minor Cannabinoids as Inhibitors of Skin Inflammation: Chemical Synthesis and Biological Evaluation
2024 A. Maiocchi, M. Fumagalli, M. Vismara, A. Blanco, U. Ciriello, G. Paladino, S. Piazza, G. Martinelli, V. Fasano, M. Dell’Agli, D. Passarella
Synthesis of α-fluorocinnamate derivatives as novel cathepsin S inhibitors with in vitro antiproliferative activity against pancreatic cancer cells
2024 A. Citarella, S. Petrella, D. Moi, A. Dimasi, T. Braga, L. Ruberto, S. Pieraccini, M. Sironi, N. Micale, T. Schirmeister, G. Damia, V. Fasano, A. Silvani, C. Giannini, D. Passarella
First Total Synthesis of Caerulomycin K: A Case Study on Selective, Multiple C-H Functionalizations of Pyridines
2024 A. Dimasi, M. Failla, A. Montoli, A. Citarella, P. Ronchi, D. Passarella, V. Fasano
A novel, glutathione-activated prodrug of pimasertib loaded in liposomes for targeted cancer therapy
2024 A. Amenta, S. Comi, M. Kravicz, S. Sesana, A. Antoniou, D. Passarella, P. Seneci, S. Pellegrino, F. Re
Recent advances in the development of {CB}1R selective probes
2023 A. Amenta, D. Caprioglio, A. Minassi, L. Panza, D. Passarella, V. Fasano, D. Imperio
Targeting Ovarian Cancer with Chalcone Derivatives: Cytotoxicity and Apoptosis Induction in HGSOC Cells
2023 E. Merve Aydin, İ.S. Canıtez, E. Colombo, S. Princiotto, D. Passarella, S. Dallavalle, M.S. Christodoulou, I. Durmaz Şahin
Structure-activity exploration of a small-molecule allosteric inhibitor of T790M/L858R double mutant EGFR
2023 F. Foschi, A. Tinivella, V. Crippa, L. Pinzi, L. Mologni, D. Passarella, G. Rastelli
Late‐Stage Functionalisation of Pyridine‐Containing Bioactive Molecules: Recent Strategies and Perspectives
2023 M. Failla, G.W. Lombardo, P. Orlando, D. Fiorito, E. Bombonato, P. Ronchi, D. Passarella, V. Fasano
2-Hydroxyoleic Acid as a Self-Assembly Inducer for Anti-Cancer Drug-Centered Nanoparticles
2023 A.I. Antoniou, G. Nordio, M. Luisa Di Paolo, E. Colombo, B. Gaffuri, L. Polito, A. Amenta, P. Seneci, L. Dalla Via, D. Perdicchia, D. Passarella
Cannabidiol as Self-Assembly Inducer for Anticancer Drug-Based Nanoparticles
2023 E. Colombo, D.A. Coppini, L. Polito, U. Ciriello, G. Paladino, M. Hyeraci, M.L. Di Paolo, G. Nordio, L. Dalla Via, D. Passarella
Synthesis and Preliminary Characterization of Putative Anle138b-Centered PROTACs against α-Synuclein Aggregation
2023 M. Pedrini, A. Iannielli, L. Meneghelli, D. Passarella, V. Broccoli, P. Seneci
Maytansinol Functionalization: Towards Useful Probes for Studying Microtubule Dynamics
2023 Z. Boiarska, H. Pérez-Peña, A. Abel, P. Marzullo, B. Álvarez-Bernad, F. Bonato, B. Santini, D. Horvath, D. Lucena-Agell, F. Vasile, M. Sironi, J.F. Díaz, A.E. Prota, S. Pieraccini, D. Passarella
Tetraphenylethylene-Based Photoluminescent Self-Assembled Nanoparticles: Preparation and Biological Evaluation
2023 E. Colombo, E.M. Aydın, İ.S. Canıtez, L. Polito, M. Penconi, A. Bossi, E. Impresari, D. Passarella, S. Dallavalle, C.M. Athanassopoulos, S. Pellegrino, I.D. Şahin, M.S. Christodoulou
Synthesis of SARS-CoV-2 Mpro Inhibitors bearing a Cinnamic Ester Warhead with In Vitro Activity against Human Coronaviruses
2023 A. Citarella, D. Moi, M. Pedrini, H. Pérez-Peña, S. Pieraccini, A. Dimasi, C. Stagno, N. Micale, T. Schirmeister, G. Sibille, G. Gribaudo, A. Silvani, C. Giannini, D. Passarella
Recent Advances in SARS-CoV-2 Main Protease Inhibitors: From Nirmatrelvir to Future Perspectives
2023 A. Citarella, A. Dimasi, D. Moi, D. Passarella, A. Scala, A. Piperno, N. Micale