FASANO, VALERIO
FASANO, VALERIO
Dipartimento di Chimica
Nirmatrelvir: from discovery to modern and alternative synthetic approaches
2024 M. Galli, F. Migliano, V. Fasano, A. Silvani, D. Passarella, A. Citarella
Nicotinic Acid Derivatives As Novel Noncompetitive α-Amylase and α-Glucosidase Inhibitors for Type 2 Diabetes Treatment
2024 A. Citarella, M. Cavinato, E. Rosini, H. Shehi, F. Ballabio, C. Camilloni, V. Fasano, A. Silvani, D. Passarella, L. Pollegioni, M. Nardini
First Total Synthesis of Caerulomycin K: A Case Study on Selective, Multiple C-H Functionalizations of Pyridines
2024 A. Dimasi, M. Failla, A. Montoli, A. Citarella, P. Ronchi, D. Passarella, V. Fasano
Synthesis of α-fluorocinnamate derivatives as novel cathepsin S inhibitors with in vitro antiproliferative activity against pancreatic cancer cells
2024 A. Citarella, S. Petrella, D. Moi, A. Dimasi, T. Braga, L. Ruberto, S. Pieraccini, M. Sironi, N. Micale, T. Schirmeister, G. Damia, V. Fasano, A. Silvani, C. Giannini, D. Passarella
Total Synthesis of an Epothilone Analogue based on the Amide‒Triazole Bioisosterism
2024 E. Colombo, D.A. Coppini, S. Borsoi, V. Fasano, R. Bucci, F. Bonato, E. Bonandi, F. Vasile, S. Pieraccini, D. Passarella
Electrochemical Synthesis of Unnatural Amino Acids Embedding 5- and 6-Membered Heteroaromatics
2024 E. Bombonato, V. Fasano, D. Pecorari, L. Fornasari, F. Castagnini, M. Marcaccio, P. Ronchi
A Green Approach to Nucleophilic Aromatic Substitutions of Nicotinic Esters in Cyrene
2024 A. Citarella, M. Cavinato, A. Amenta, M. Nardini, A. Silvani, D. Passarella, V. Fasano
Minor Cannabinoids as Inhibitors of Skin Inflammation: Chemical Synthesis and Biological Evaluation
2024 A. Maiocchi, M. Fumagalli, M. Vismara, A. Blanco, U. Ciriello, G. Paladino, S. Piazza, G. Martinelli, V. Fasano, M. Dell’Agli, D. Passarella
Late‐Stage Functionalisation of Pyridine‐Containing Bioactive Molecules: Recent Strategies and Perspectives
2023 M. Failla, G.W. Lombardo, P. Orlando, D. Fiorito, E. Bombonato, P. Ronchi, D. Passarella, V. Fasano
De Novo Synthesis of Dihydrobenzofurans and Indolines and Its Application to a Modular, Asymmetric Synthesis of Beraprost
2023 Z. Wang, S.H. Bennett, B. Kicin, C. Jing, J.A. Pradeilles, K. Thai, J.R. Smith, P. David Bacoş, V. Fasano, C.M. Saunders, V.K. Aggarwal
Recent advances in the development of {CB}1R selective probes
2023 A. Amenta, D. Caprioglio, A. Minassi, L. Panza, D. Passarella, V. Fasano, D. Imperio
Automated stereocontrolled assembly-line synthesis of organic molecules
2022 V. Fasano, R.C. Mykura, J.M. Fordham, J.J. Rogers, B. Banecki, A. Noble, V.K. Aggarwal
Stereoselective Synthetic Strategies to (-)-Cannabidiol
2022 A. Maiocchi, J. Barbieri, V. Fasano, D. Passarella
Origin of stereocontrol in the Matteson reaction: Importance of attractive electrostatic interactions
2021 V. Fasano, V.K. Aggarwal
Highly Diastereoselective Strain-Increase Allylborations: Rapid Access to Alkylidenecyclopropanes and Alkylidenecyclobutanes
2021 D.P. Hari, R. Madhavachary, V. Fasano, J. Haire, V.K. Aggarwal
Direct Observation of Reactive Intermediates by Time-Resolved Spectroscopy Unravels the Mechanism of a Radical-Induced 1,2-Metalate Rearrangement
2021 L. Lewis-Borrell, M. Sneha, I.P. Clark, V. Fasano, A. Noble, V.K. Aggarwal, A.J. Orr-Ewing
How Big is the Pinacol Boronic Ester as a Substituent?
2020 V. Fasano, A.W. Mcford, C.P. Butts, B.S.L. Collins, N. Fey, R.W. Alder, V.K. Aggarwal
Synthesis, Stability, and Biological Studies of Fluorinated Analogues of Thromboxane A2
2020 C. Jing, S. Mallah, E. Kriemen, S.H. Bennett, V. Fasano, A.J.J. Lennox, I. Hers, V.K. Aggarwal
Difunctionalization of C−C σ‑Bonds Enabled by the Reaction of Bicyclo[1.1.0]butyl Boronate Complexes with Electrophiles: Reaction development, scope, and stereochemical origins
2020 S.H. Bennett, A. Fawcett, E.H. Denton, T. Biberger, V. Fasano, N. Winter, V.K. Aggarwal
Ring-Expansion Induced 1,2-Metalate Rearrangements: Highly Diastereoselective Synthesis of Cyclobutyl Boronic Esters
2020 D.P. Hari, J.C. Abell, V. Fasano, V.K. Aggarwal