GRAZIOSO, GIOVANNI
GRAZIOSO, GIOVANNI
Dipartimento di Scienze Farmaceutiche
(-)-HIP-A and (+)-HIP-B: investigation of the pharmacological profile and potential therapeutic applications
2007 P. Conti, A. Pinto, L. Tamborini, G. Grazioso, S. Colleoni, M. Gobbi, T. Mennini
Ago-allosteric modulation of nicotinic alpha7 receptors : a mechanistic insight by metadynamics and essential dynamics
2014 G. Grazioso
Agonisti nicotinici selettivi nel trattamento di patologie del Sistema Nervoso Centrale
2007 C. De Micheli, M. De Amici, C. Dallanoce, G. Grazioso, L. Rizzi, P. Magrone, C. Matera
Alkene Epoxidations Mediated by Mn-Salen Macrocyclic Catalysts
2021 A. Pappalardo, F.P. Ballistreri, R.M. Toscano, M.A. Chiacchio, L. Legnani, G. Grazioso, L. Veltri, G. Trusso Sfrazzetto
Allosteric modulation of alpha7 nicotinic receptors : mechanistic insight through metadynamics and essential dynamics
2015 G. Grazioso, J. Sgrignani, R. Capelli, C. Matera, C. Dallanoce, M. De Amici, A. Cavalli
Alpha7 nicotinic acetylcholine receptor agonists: prediction of their binding affinity through a molecular mechanics poisson-boltzmann surface area approach
2008 G. Grazioso, A. Cavalli, M. De Amici, M. Recanatini, C. De Micheli
Analytical, computational and formulation studies on TPGS as P-gp inhibitor
2015 M.D. Del Curto, C. Bolchi, A. Foppoli, L. Fumagalli, F. Selmin, G. Grazioso, L. Palugan
Application of the Ugi reaction with multiple amino acid-derived components : synthesis and conformational evaluation of piperazine-based minimalist peptidomimetics
2015 M. Stucchi, S. Cairati, R. Cetin Atalay, M. Christodoulou, G. Grazioso, G. Pescitelli, A. Silvani, D.C. Yildirim, G. Lesma
Bifunctional compounds targeting both D2 and non-α7 nACh receptors: design, synthesis and pharmacological characterization
2015 C. Matera, L. Pucci, C. Fiorentini, S. Fucile, C. Missale, G. Grazioso, F. Clementi, M. Zoli, M. De Amici, C. Gotti, C. Dallanoce
Bioactive cyclization optimizes the affinity of a proprotein convertase subtilisin/kexin type 9 (PCSK9) peptide inhibitor
2021 B.J. Tombling, C. Lammi, N. Lawrence, E.K. Gilding, G. Grazioso, D.J. Craik, C.K. Wang
Biological Characterization of Computationally Designed Analogs of peptide TVFTSWEEYLDWV (Pep2-8) with Increased PCSK9 Antagonistic Activity
2019 C. Lammi, J. Sgrignani, A. Arnoldi, G. Grazioso
Computational approaches in the rational design of improved carbonyl quenchers : focus on histidine containing dipeptides
2016 G. Vistoli, M. Colzani, A. Mazzolari, D.D. Maddis, G. Grazioso, A. Pedretti, M. Carini, G. Aldini
Computational Design and Biological Evaluation of Analogs of Lupin Peptide P5 Endowed with Dual PCSK9/HMG-CoAR Inhibiting Activity
2022 C. Lammi, E. Fassi, J. Li, M. Bartolomei, G. Benigno, G. Roda, A. Arnoldi, G. Grazioso
Computational Design, Synthesis, and Biophysical Evaluation of β-Amido Boronic Acids as SARS-CoV-2 Mpro Inhibitors
2023 E.M.A. Fassi, M. Manenti, A. Citarella, M. Dei Cas, S. Casati, N. Micale, T. Schirmeister, G. Roda, A. Silvani, G. Grazioso
COMPUTATIONAL INVESTIGATION ON SUBSTRATE UPTAKE AND RELEASE IN A GLUTAMATE TRANSPORTER
2012 G. Grazioso, V. Limongelli, D. Branduardi, E. Novellino, C. De Micheli, A. Cavalli, M. Parrinello
Computationally Driven Structure Optimization, Synthesis, and Biological Evaluation of Imidazole-Based Proprotein Convertase Subtilisin/Kexin 9 (PCSK9) Inhibitors
2019 C. Lammi, J. Sgrignani, A. Arnoldi, G. Lesma, C. Spatti, A. Silvani, G. Grazioso
Covalent docking of selected boron-based serine beta-lactamase inhibitors
2015 J. Sgrignani, B. Novati, G. Colombo, G. Grazioso
Design and synthesis of selective ligands targeting different nAChR subtypes
2014 M. Quadri, C. Matera, G. Grazioso, M. De Amici, C. Dallanoce
Design of Cyclopentaisoxazoline Amino Acids as Conformationally Constrained Agonists at Glutamate Receptors
2003 P. Conti, M. De Amici, G. Grazioso, G. Roda, T.B. Stensbøl, H. Bräuner-Osborne, U. Madsen, L. Toma, C. De Micheli
Design of novel α7-subtype-preferring nicotinic acetylcholine receptor agonists: application of docking and MM-PBSA computational approaches, synthetic and pharmacological studies
2009 G. Grazioso, D.Y. Pomè, C. Matera, F. Frigerio, L. Pucci, C. Gotti, C. Dallanoce, M. De Amici