FASSI, ENRICO MARIO ALESSANDRO
FASSI, ENRICO MARIO ALESSANDRO
Dipartimento di Scienze Farmaceutiche
Insights into the catalytic mechanism of formate dehydrogenases from different microbial sources
2026 L. Legnani, M. Gargiulo, E. Lio, E.M.A. Fassi, G. Grazioso, M.A. Chiacchio, B. Binay, S. Brocca, F. Secundo
Insights on Zosteric Acid Analogues Activity Against Candida albicans Biofilm Formation
2025 C. Catto', E.M.A. Fassi, G. Grazioso, A. Gelain, S. Villa, F. Cappitelli
Design and synthesis of CD70 inhibitors: a potential way for the treatment of ulcerative colitis
2025 M. Galli, A. Silvani, G. Grazioso, E.G. Milano, E.M.A. Fassi, M. Bramuzzo, A. Muzzo, G. Stocco, M. Lucafò
Modulatori Fotosensibili dell’adesione batterica: una nuova strategia per ridurre l’antibiotico-resistenza
2025 A. Colleoni, G. Tempra, S. Bhattacharya, E.M.A. Fassi, M. De Amici, G. Grazioso, R. Castagna, E. Parisini, C. Matera
Spatiotemporal Control of Bacterial Adhesion via Light-Responsive Modulators
2025 A. Colleoni, G. Tempra, S. Bhattacharya, E.M.A. Fassi, M. De Amici, G. Grazioso, R. Castagna, E. Parisini, C. Matera
Support Vector Machine Identification of Small Molecule Binders to an Understudied Allosteric Site of SARS‐CoV‐2 Mpro for Next‐Generation PROTAC‐Based Therapeutics
2025 E.M.A. Fassi, N. Mekni, M. Albani, S. Maehrlein, A.C. Weldert, T. Schirmeister, T. Langer, G. Grazioso
Light-Responsive Modulators of Bacterial Cell Adhesion Proteins: a Novel Strategy against AMR?
2025 A. Colleoni, G. Tempra, S. Bhattacharya, E.M.A. Fassi, M. De Amici, G. Grazioso, R. Castagna, E. Parisini, C. Matera
FYCO1 Peptide Analogs: Design and Characterization of Autophagy Inhibitors as Co-Adjuvants in Taxane Chemotherapy of Prostate Cancer
2025 E.M.A. Fassi, R.M. Moretti, M. Montagnani Marelli, M. Garofalo, A. Gori, C. Pesce, M. Albani, E.G. Milano, J. Sgrignani, A. Cavalli, G. Grazioso
Nature‐Inspired Compounds Targeting Escherichia coli WrbA as Biofilm‐Modulating Agents: Computational Design, Synthesis, and Biological Evaluation
2025 M. Mori, E.M.A. Fassi, F. Villa, E.G. Milano, F. Forlani, F. Cappitelli, A. Ratti, F. Meneghetti, G. Roda, G. Grazioso, S. Villa
Enhancing the activity of γ-hydroxy lactone derivatives as innovative peroxisome proliferator-activated receptor γ non-agonists inhibiting cyclin-dependent kinase 5-mediated phosphorylation
2025 G. Cazzaniga, D. Capelli, R. Montanari, E.M.A. Fassi, G. Grazioso, A. Tresoldi, F. Rinaldi, E. Calleri, I. Bassanini, S. Romeo, M. Garofalo, M. Mori, F. Meneghetti, S. Villa
A potent nonapeptide inhibitor for the CXCL12/HMGB1 heterocomplex: A computational and experimental approach
2025 E.M.A. Fassi, E. Pirani, V. Cecchinato, A. Cavalli, G. Roda, M. Uguccioni, J. Sgrignani, G. Grazioso
Computational Design of Novel Cyclic Peptides Endowed with Autophagy-Inhibiting Activity on Cancer Cell Lines
2024 M. Albani, E.M.A. Fassi, R.M. Moretti, M. Garofalo, M. Montagnani Marelli, G. Roda, J. Sgrignani, A. Cavalli, G. Grazioso
High‐throughput peptide array analysis and computational techniques for serological profiling of flavivirus infections: Implications for diagnostics and vaccine development
2024 M. Bombaci, E.M.A. Fassi, A. Gobbini, D. Mileto, I. Cassaniti, E. Pesce, E. Casali, A. Mancon, J. Sammartino, A. Ferrari, E. Percivalle, R. Grande, E. Marchisio, M.R. Gismondo, S. Abrignani, F. Baldanti, G. Colombo, R. Grifantini
Towards a safe treatment of Insulin Resistance: γ-hydroxy lactone-based derivatives as PPARγ non-agonists
2024 G. Cazzaniga, M. Mori, D. Capelli, R. Montanari, A. Laghezza, F. Loiodice, E.M.A. Fassi, G. Grazioso, F. Meneghetti, S. Villa
PCSK9 inhibitors: a patent review 2018-2023
2024 E.M.A. Fassi, A. Citarella, M. Albani, E.G. Milano, L. Legnani, C. Lammi, A. Silvani, G. Grazioso
Novel Non-peptide Uracil-derived Human Gonadotropin-Releasing Hormone Receptor Antagonists
2024 S. Ciceri, E.M.A. Fassi, V. Vezzoli, M. Bonomi, D. Colombo, P. Ferraboschi, G. Grazioso, P. Grisenti, S. Villa, C. Castellano, F. Meneghetti
Elagolix Sodium Salt and Its Synthetic Intermediates: A Spectroscopic, Crystallographic, and Conformational Study
2023 S. Ciceri, D.R. Colombo, E.M.A. Fassi, P. Ferraboschi, G. Grazioso, P. Grisenti, M. Iannone, C. Castellano, F. Meneghetti
Unlocking the Antibiofilm Potential of Natural Compounds by Targeting the NADH:quinone Oxidoreductase WrbA
2023 A. Ratti, E.M.A. Fassi, F. Forlani, M. Zangrossi, M. Mori, F. Cappitelli, G. Roda, S. Villa, F. Villa, G. Grazioso
Computational Design, Synthesis, and Biophysical Evaluation of β-Amido Boronic Acids as SARS-CoV-2 Mpro Inhibitors
2023 E.M.A. Fassi, M. Manenti, A. Citarella, M. Dei Cas, S. Casati, N. Micale, T. Schirmeister, G. Roda, A. Silvani, G. Grazioso
γ-HYDROXY LACTONE BASED PPARγ NON-AGONISTS AS SAFE AND INNOVATIVE ANTI-DIABETIC AGENTS
2023 G. Cazzaniga, M. Mori, D. Capelli, R. Montanari, A. Laghezza, F. Loiodice, I. Bassanini, S. Romeo, E.M.A. Fassi, G. Grazioso, M. Quaglia, F. Meneghetti, S. Villa