FASSI, ENRICO MARIO ALESSANDRO

FASSI, ENRICO MARIO ALESSANDRO  

Dipartimento di Scienze Farmaceutiche  

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Titolo Data di pubblicazione Autori Tipo File Abstract
A potent nonapeptide inhibitor for the CXCL12/HMGB1 heterocomplex: A computational and experimental approach 2025 Fassi, Enrico Mario AlessandroRoda, GabriellaGrazioso, Giovanni + Article (author) -
Enhancing the activity of γ-hydroxy lactone derivatives as innovative peroxisome proliferator-activated receptor γ non-agonists inhibiting cyclin-dependent kinase 5-mediated phosphorylation 2025 Cazzaniga, GiuliaFassi, Enrico Mario AlessandroGrazioso, GiovanniTresoldi, AndreaBassanini, IvanRomeo, SergioMori, MatteoMeneghetti, FiorellaVilla, Stefania + Article (author) -
Exploiting the Potential of Computational Approaches in Medicinal Chemistry: CADD of Novel eIF6 Binders for the Development of anti-HCC PROTACs 2025 Alessio ColleoniEnrico M. A. FassiA. MiluzioGiorgia TempraMarco AlbaniMarco De AmiciGiovanni GraziosoStefano BiffoCarlo Matera Conference Object -
Towards a safe treatment of Insulin Resistance: γ-hydroxy lactone-based derivatives as PPARγ non-agonists 2024 G. CazzanigaM. MoriE. M. A. FassiG. GraziosoF. MeneghettiS. Villa + Conference Object -
Targeted degraders of eIF6: a novel strategy to remodulate liver pathological lipidic metabolism 2024 Alessio ColleoniEnrico M. A. FassiAnnarita MiluzioMarco AlbaniMarco De AmiciGiovanni GraziosoStefano BiffoCarlo Matera + Conference Object -
Tackling Hepatocellular Carcinoma with Targeted Degraders of eIF6 2024 A. ColleoniEnrico M. A. FassiA. MiluzioM. AlbaniM. De AmiciG. GraziosoS. BiffoC. Matera + Conference Object -
Novel Non-peptide Uracil-derived Human Gonadotropin-Releasing Hormone Receptor Antagonists 2024 Ciceri, SamueleFassi, Enrico M. A.Vezzoli, ValeriaBonomi, MarcoColombo, DiegoFerraboschi, PatriziaGrazioso, GiovanniVilla, StefaniaCastellano, CarloMeneghetti, Fiorella + Article (author) -
PCSK9 inhibitors: a patent review 2018-2023 2024 Fassi, Enrico Mario AlessandroCitarella, AndreaAlbani, MarcoMilano, Erica GinevraLegnani, LauraLammi, CarmenSilvani, AlessandraGrazioso, Giovanni Article (author) -
Computational Design of Novel Cyclic Peptides Endowed with Autophagy-Inhibiting Activity on Cancer Cell Lines 2024 Albani, MarcoFassi, Enrico Mario AlessandroMoretti, Roberta ManuelaMontagnani Marelli, MarinaRoda, GabriellaGrazioso, Giovanni + Article (author) -
High‐throughput peptide array analysis and computational techniques for serological profiling of flavivirus infections: Implications for diagnostics and vaccine development 2024 Fassi, Enrico Mario AlessandroMileto, DavideCassaniti, IrenePesce, ElisaMancon, AlessandroGismondo, Maria RitaAbrignani, Sergio + Article (author) -
Insights on the atropisomeric properties of elagolix and its derivatives 2023 Samuele CiceriDiego ColomboEnrico M. A. FassiPatrizia FerraboschiGiovanni GraziosoFiorella Meneghetti + Conference Object -
A new class of GnRH receptor modulators endowed with atropisomerism 2023 Samuele CiceriDiego ColomboEnrico M. A. FassiPatrizia FerraboschiGiovanni GraziosoFiorella Meneghetti + Conference Object -
Mechanistic Insights into the Antibiofilm Mode of Action of Ellagic Acid 2023 Ratti, AlessandroFassi, Enrico M. A.Forlani, FabioMori, MatteoVilla, FedericaCappitelli, FrancescaRoda, GabriellaVilla, StefaniaGrazioso, Giovanni + Article (author) -
COMPUTATIONAL DESIGN OF PEPTIDES AND PEPTIDOMIMETICS AS POTENTIAL THERAPEUTIC AGENTS TO SATISFY PRESSING MEDICAL NEEDS 2023 FASSI, ENRICO MARIO ALESSANDRO Doctoral Thesis -
Natural and nature-inspired compounds targeting E. coli WrbA as antibiofilm agents: computational studies, synthesis, and biological evaluation 2023 Mori, M.Villa, S.Ratti, A.Meneghetti, F.Roda, G.Gelain, A.Villa F.Fassi, E. M. A.Forlani, F.Grazioso, G. Conference Object -
γ-hidroxy-lactone derivatives as ppar-γ non-agonists blocking cdk5-mediated phosporylation for a safer anti-diabetic treatment 2023 G. CazzanigaM. MoriI. BassaniniS. RomeoE. M. A. FassiM. QuagliaG. GraziosoF. MeneghettiS. Villa + Conference Object -
γ-HYDROXY LACTONE BASED PPARγ NON-AGONISTS AS SAFE AND INNOVATIVE ANTI-DIABETIC AGENTS 2023 G. CazzanigaM. MoriI. BassaniniS. RomeoE. M. A. FassiG. GraziosoM. QuagliaF. MeneghettiS. Villa + Conference Object -
γ-HYDROXY LACTONE BASED PPARγ NON-AGONISTS AS SAFE AND INNOVATIVE ANTI-DIABETIC AGENTS. 2023 G. CazzanigaM. MoriI. BassaniniS. RomeoE. M. A. FassiG. GraziosoM. QuagliaF. MeneghettiS. Villa + Conference Object -
Computational Design, Synthesis, and Biological Evaluation of Diimidazole Analogues Endowed with Dual PCSK9/HMG-CoAR-Inhibiting Activity 2023 Carmen LammiEnrico M. A. FassiMarco ManentiJianqiang LiGabriella RodaMarina CameraAlessandra SilvaniGiovanni Grazioso + Article (author) -
Computational Design, Synthesis, and Biophysical Evaluation of β-Amido Boronic Acids as SARS-CoV-2 Mpro Inhibitors 2023 Fassi, Enrico M. A.Manenti, MarcoCitarella, AndreaDei Cas, MicheleCasati, SaraRoda, GabriellaSilvani, AlessandraGrazioso, Giovanni + Article (author) -