FASSI, ENRICO MARIO ALESSANDRO
FASSI, ENRICO MARIO ALESSANDRO
Dipartimento di Scienze Farmaceutiche
Protein language model-generated enzyme sequences exhibit high stability in molecular dynamics simulations
2026 E.M.A. Fassi, M. Nicolini, E. Saitto, G. Valentini, E. Casiraghi, G. Grazioso
Insights into the catalytic mechanism of formate dehydrogenases from different microbial sources
2026 L. Legnani, M. Gargiulo, E. Lio, E.M.A. Fassi, G. Grazioso, M.A. Chiacchio, B. Binay, S. Brocca, F. Secundo
Finenzyme-generated enzymes with predicted structures (ESMfold)
2026 M. Nicolini, E. Fassi, G. Valentini, E. Casiraghi, G. Grazioso
Targeting Pseudomonas aeruginosa LecB with Photoswitchable Glycomimetic Ligands
2026 A. Colleoni, S. Bhattacharya, G. Tempra, E.M.A. Fassi, M. De Amici, G. Grazioso, R. Castagna, E. Parisini, C. Matera
Development of In-Cell Self-Assembly Proteolysis Targeting Chimeras Exploiting the Biorthogonal Reaction Between Vinyl Boronic Acids and 1,2,4,5-Tetrazines
2026 M. Galli, L. Passarelli, E. Fassi, G. Grazioso, D. Passarella, A. Silvani
Synthesis of Self-Assembling Proteolysis Targeting Chimeras Based on Biorthogonal Reactions
2026 M. Galli, L. Passarelli, A. Silvani, G. Grazioso, E. Fassi
PCSK9 inhibitors: an updated patent review 2024–2025
2026 E.M.A. Fassi, M. Albani, L. D'Adduzio, E.G. Milano, C. Lammi, G. Grazioso
Breakable Organosilica Nanocapsules for the Intracellular Delivery of a Peptide With Promising Anti‐Breast Cancer Activity
2026 S. Mathlouthi, A. Ajò, E.M.A. Fassi, A. Cagnotto, A. Fragassi, C. Pesce, M. Garofalo, L. De Cola, G. Grazioso
Design, synthesis and characterization of novel potential TAU-degraders
2026 G. Tempra, E.M.A. Fassi, G. Grazioso, P. Seneci, D. Passarella
A nicotinic-dopaminergic hybrid probe enhances D2-like autoreceptor-mediated inhibition of dopamine release
2026 C. Matera, M. Grilli, L. Pucci, E.M.A. Fassi, S. Fucile, M. Marchi, C. Fiorentini, F. Clementi, M. Zoli, C. Dallanoce, G. Grazioso, M. De Amici, C. Gotti
Structure-guided design of an LC3B-targeting PNA oligomer modulating autophagy and LC3B-mediated mRNA decay
2026 M. Albani, E.M.A. Fassi, A. Romanelli, M. Montagnani Marelli, M. Garofalo, G. Roda, R.M. Moretti, G. Grazioso
Spatiotemporal Control of Bacterial Adhesion via Light-Responsive Modulators
2025 A. Colleoni, G. Tempra, S. Bhattacharya, E.M.A. Fassi, M. De Amici, G. Grazioso, R. Castagna, E. Parisini, C. Matera
Design and synthesis of CD70 inhibitors: a potential way for the treatment of ulcerative colitis
2025 M. Galli, A. Silvani, G. Grazioso, E.G. Milano, E.M.A. Fassi, M. Bramuzzo, A. Muzzo, G. Stocco, M. Lucafò
Support Vector Machine Identification of Small Molecule Binders to an Understudied Allosteric Site of SARS‐CoV‐2 Mpro for Next‐Generation PROTAC‐Based Therapeutics
2025 E.M.A. Fassi, N. Mekni, M. Albani, S. Maehrlein, A.C. Weldert, T. Schirmeister, T. Langer, G. Grazioso
A potent nonapeptide inhibitor for the CXCL12/HMGB1 heterocomplex: A computational and experimental approach
2025 E.M.A. Fassi, E. Pirani, V. Cecchinato, A. Cavalli, G. Roda, M. Uguccioni, J. Sgrignani, G. Grazioso
Enhancing the activity of γ-hydroxy lactone derivatives as innovative peroxisome proliferator-activated receptor γ non-agonists inhibiting cyclin-dependent kinase 5-mediated phosphorylation
2025 G. Cazzaniga, D. Capelli, R. Montanari, E.M.A. Fassi, G. Grazioso, A. Tresoldi, F. Rinaldi, E. Calleri, I. Bassanini, S. Romeo, M. Garofalo, M. Mori, F. Meneghetti, S. Villa
Light-Responsive Modulators of Bacterial Cell Adhesion Proteins: a Novel Strategy against AMR?
2025 A. Colleoni, G. Tempra, S. Bhattacharya, E.M.A. Fassi, M. De Amici, G. Grazioso, R. Castagna, E. Parisini, C. Matera
Modulatori Fotosensibili dell’adesione batterica: una nuova strategia per ridurre l’antibiotico-resistenza
2025 A. Colleoni, G. Tempra, S. Bhattacharya, E.M.A. Fassi, M. De Amici, G. Grazioso, R. Castagna, E. Parisini, C. Matera
Nature‐Inspired Compounds Targeting Escherichia coli WrbA as Biofilm‐Modulating Agents: Computational Design, Synthesis, and Biological Evaluation
2025 M. Mori, E.M.A. Fassi, F. Villa, E.G. Milano, F. Forlani, F. Cappitelli, A. Ratti, F. Meneghetti, G. Roda, G. Grazioso, S. Villa
FYCO1 Peptide Analogs: Design and Characterization of Autophagy Inhibitors as Co-Adjuvants in Taxane Chemotherapy of Prostate Cancer
2025 E.M.A. Fassi, R.M. Moretti, M. Montagnani Marelli, M. Garofalo, A. Gori, C. Pesce, M. Albani, E.G. Milano, J. Sgrignani, A. Cavalli, G. Grazioso