DIMASI, ALESSANDRO
DIMASI, ALESSANDRO
Dipartimento di Chimica
Synthesis and Multitarget Inhibitory Effect of Indole-Based Ethyl Cinnamate Derivatives against SARS-CoV-2 Mpro and Cathepsins for Broad-Spectrum Anti-Coronavirus Activity
2025 A. Citarella, G. Sibile, D. Moi, A. Dimasi, T. Braga, L. Dal Col, L. Ruberto, S. Pieraccini, M. Sironi, N. Micale, T. Schirmeister, V. Fasano, A. Silvani, C. Giannini, G. Gribaudo, D. Passarella
Mechanistic insights into the base-mediated deuteration of pyridyl phosphonium and ammonium salts
2025 A. Montoli, A. Dimasi, M. Guarnaccia, A. Citarella, P. Ronchi, D. Blasi, S. Rossi, D. Passarella, V. Fasano
Metal‐Free, Selective Ortho‐Deuteration of N‐Heterocyclic Oxides
2025 A. Montoli, A. Dimasi, A. Citarella, P. Ronchi, D. Passarella, V. Fasano
Synthesis and multitarget inhibitory effect of indole-based ethyl cinnamate derivatives against SARS-CoV-2 Mpro and cathepsins for broad-spectrum anti-coronavirus activity
2025 A. Citarella, G. Sibille, D. Moi, A. Dimasi, T. Braga, L.D. Col, L. Ruberto, S. Pieraccini, M. Sironi, N. Micale, T. Schirmeister, V. Fasano, A. Silvani, C. Giannini, G. Gribaudo, D. Passarella
Synthesis of α-fluorocinnamate derivatives as novel cathepsin S inhibitors with in vitro antiproliferative activity against pancreatic cancer cells
2024 A. Citarella, S. Petrella, D. Moi, A. Dimasi, T. Braga, L. Ruberto, S. Pieraccini, M. Sironi, N. Micale, T. Schirmeister, G. Damia, V. Fasano, A. Silvani, C. Giannini, D. Passarella
First Total Synthesis of Caerulomycin K: A Case Study on Selective, Multiple C-H Functionalizations of Pyridines
2024 A. Dimasi, M. Failla, A. Montoli, A. Citarella, P. Ronchi, D. Passarella, V. Fasano
Recent Advances in SARS-CoV-2 Main Protease Inhibitors: From Nirmatrelvir to Future Perspectives
2023 A. Citarella, A. Dimasi, D. Moi, D. Passarella, A. Scala, A. Piperno, N. Micale