SILVANI, ALESSANDRA
SILVANI, ALESSANDRA
Dipartimento di Chimica
Synthesis and Multitarget Inhibitory Effect of Indole-Based Ethyl Cinnamate Derivatives against SARS-CoV-2 Mpro and Cathepsins for Broad-Spectrum Anti-Coronavirus Activity
2025 A. Citarella, G. Sibile, D. Moi, A. Dimasi, T. Braga, L. Dal Col, L. Ruberto, S. Pieraccini, M. Sironi, N. Micale, T. Schirmeister, V. Fasano, A. Silvani, C. Giannini, G. Gribaudo, D. Passarella
Synthesis and multitarget inhibitory effect of indole-based ethyl cinnamate derivatives against SARS-CoV-2 Mpro and cathepsins for broad-spectrum anti-coronavirus activity
2025 A. Citarella, G. Sibille, D. Moi, A. Dimasi, T. Braga, L.D. Col, L. Ruberto, S. Pieraccini, M. Sironi, N. Micale, T. Schirmeister, V. Fasano, A. Silvani, C. Giannini, G. Gribaudo, D. Passarella
Structure-Based Discovery of Hsp90/HDAC6 Dual Inhibitors Targeting Aggressive Prostate Cancer
2025 A. Citarella, S. Belluti, D. Bonanni, D. Moi, I. Piccinini, A. Rinaldi, C. Papulino, R. Benedetti, L. Cuoghi, S.D. Ciolo, A. Silvani, L. Altucci, L. Pinzi, S. Franchini, D. Passarella, C. Sorbi, C. Giannini, C. Imbriano, G. Rastelli
Sustainable Synthesis of 1,2,3‐Triazoles using Cyrene as a Biodegradable Solvent in Click Chemistry
2025 A. Citarella, A. Fiori, A. Silvani, D. Passarella, V. Fasano
Design, synthesis and characterization of aryl bis-guanyl hydrazones as RNA binders of C9orf72 G4C2 extended repeats
2025 A. Maiocchi, M. Pedrini, V. Ferrari, A.S. Assunçao Carreira, V.M. D'Amore, F. Santoro, A. Di Porzio, M. Bosetti, R. Cristofani, A. Silvani, D. Brancaccio, L. Marinelli, F.S. Di Leva, A. Provenzani, A. Poletti, P. Seneci
Modular Symmetric Ligands for Selective Recognition of Cancer-Relevant G-Quadruplexes
2024 C. Platella, A. Citarella, M. Manenti, G. Spinelli, R. Gaglione, A. Arciello, C. Riccardi, D. Musumeci, D. Montesarchio, C. Giannini, A. Silvani
Poly(alditol sebacate)-PLA copolymers: enhanced degradability and tunable surface properties
2024 S. Gazzotti, M. Hakkarainen, C.A. Pagnacco, M. Manenti, A. Silvani, H. Farina, L. Arnaboldi, M.A. Ortenzi
PCSK9 inhibitors: a patent review 2018-2023
2024 E.M.A. Fassi, A. Citarella, M. Albani, E.G. Milano, L. Legnani, C. Lammi, A. Silvani, G. Grazioso
Nirmatrelvir: from discovery to modern and alternative synthetic approaches
2024 M. Galli, F. Migliano, V. Fasano, A. Silvani, D. Passarella, A. Citarella
Alkene carboamination/oxidative denitrogenation of 3-allyl-3-hydrazinylindolin-2-ones: one-pot entry to spirocyclopropyloxindoles
2024 M. Manenti, T. Villa, G. Macetti, A. Silvani
A Green Approach to Nucleophilic Aromatic Substitutions of Nicotinic Esters in Cyrene
2024 A. Citarella, M. Cavinato, A. Amenta, M. Nardini, A. Silvani, D. Passarella, V. Fasano
Nicotinic Acid Derivatives As Novel Noncompetitive α-Amylase and α-Glucosidase Inhibitors for Type 2 Diabetes Treatment
2024 A. Citarella, M. Cavinato, E. Rosini, H. Shehi, F. Ballabio, C. Camilloni, V. Fasano, A. Silvani, D. Passarella, L. Pollegioni, M. Nardini
Chemical modifications of aromatic scaffolds for the development of new G4 ligands
2024 S. Di Ciolo, B. Airoldi, L.C.M. Pariani, C.F. Morelli, C. Giannini, A. Silvani, D. Malpicci, E. Cariati, E. Lucenti, C. Platella, D. Musumeci, R. Gaglione, A. Arciello, D. Montesarchio
Innovative molecular platforms for G-quadruplex stabilizatioN
2024 S. Di Ciolo, B. Airoldi, L.C.M. Pariani, C.F. Morelli, C. Giannini, A. Silvani, D. Malpicci, E. Cariati, E. Lucenti, C. Platella, D. Musumeci, R. Gaglione, A. Arciello, D. Montesarchio
Innovative molecular platforms for G-quadruplex stabilization
2024 S. Di Ciolo, B. Airoldi, L.C.M. Pariani, C.F. Morelli, C. Giannini, A. Silvani, D. Malpicci, E. Cariati, E. Lucenti, C. Platella, D. Musumeci, R. Gaglione, A. Arciello, D. Montesarchio
Synthesis of α-fluorocinnamate derivatives as novel cathepsin S inhibitors with in vitro antiproliferative activity against pancreatic cancer cells
2024 A. Citarella, S. Petrella, D. Moi, A. Dimasi, T. Braga, L. Ruberto, S. Pieraccini, M. Sironi, N. Micale, T. Schirmeister, G. Damia, V. Fasano, A. Silvani, C. Giannini, D. Passarella
Computational Design, Synthesis, and Biological Evaluation of Diimidazole Analogues Endowed with Dual PCSK9/HMG-CoAR-Inhibiting Activity
2023 C. Lammi, E.M.A. Fassi, M. Manenti, M. Brambilla, M. Conti, J. Li, G. Roda, M. Camera, A. Silvani, G. Grazioso
Computational Design, Synthesis, and Biophysical Evaluation of β-Amido Boronic Acids as SARS-CoV-2 Mpro Inhibitors
2023 E.M.A. Fassi, M. Manenti, A. Citarella, M. Dei Cas, S. Casati, N. Micale, T. Schirmeister, G. Roda, A. Silvani, G. Grazioso
Mechanistic insights of the copper(I)-catalysed reaction between chlorohydrazones and terminal alkynes
2023 A. Ponti, A. Silvani, G. Molteni
Synthesis of SARS-CoV-2 Mpro Inhibitors bearing a Cinnamic Ester Warhead with In Vitro Activity against Human Coronaviruses
2023 A. Citarella, D. Moi, M. Pedrini, H. Pérez-Peña, S. Pieraccini, A. Dimasi, C. Stagno, N. Micale, T. Schirmeister, G. Sibille, G. Gribaudo, A. Silvani, C. Giannini, D. Passarella