RUBERTO, LORENZO
RUBERTO, LORENZO
Dipartimento di Chimica
Synthesis and Multitarget Inhibitory Effect of Indole-Based Ethyl Cinnamate Derivatives against SARS-CoV-2 Mpro and Cathepsins for Broad-Spectrum Anti-Coronavirus Activity
2025 A. Citarella, G. Sibile, D. Moi, A. Dimasi, T. Braga, L. Dal Col, L. Ruberto, S. Pieraccini, M. Sironi, N. Micale, T. Schirmeister, V. Fasano, A. Silvani, C. Giannini, G. Gribaudo, D. Passarella
Synthesis and multitarget inhibitory effect of indole-based ethyl cinnamate derivatives against SARS-CoV-2 Mpro and cathepsins for broad-spectrum anti-coronavirus activity
2025 A. Citarella, G. Sibille, D. Moi, A. Dimasi, T. Braga, L.D. Col, L. Ruberto, S. Pieraccini, M. Sironi, N. Micale, T. Schirmeister, V. Fasano, A. Silvani, C. Giannini, G. Gribaudo, D. Passarella
Design, synthesis and in vitro validation of bivalent binders of SARS-CoV-2 spike protein: Obeticholic, betulinic and glycyrrhetinic acids as building blocks
2025 M. Pedrini, L. Pozzi, F. Sacchi, A. Citarella, V. Fasano, P. Seneci, S. Pieraccini, L. Ruberto, H. Perez Peña, A. Garzino-Demo, A. Vitiello, L. Sernicola, A. Borsetti, A. Calistri, C. Parolin, D. Passarella
Synthesis of α-fluorocinnamate derivatives as novel cathepsin S inhibitors with in vitro antiproliferative activity against pancreatic cancer cells
2024 A. Citarella, S. Petrella, D. Moi, A. Dimasi, T. Braga, L. Ruberto, S. Pieraccini, M. Sironi, N. Micale, T. Schirmeister, G. Damia, V. Fasano, A. Silvani, C. Giannini, D. Passarella
Development of docking protocol for small molecules on tubulin
2024 L. Ruberto, M. Sironi, S. Pieraccini