GIANNINI, CLELIA
GIANNINI, CLELIA
Dipartimento di Chimica
Combining Cyclic Triimidazo Triazine Core With Ethynyl‐N‐Methyl‐Pyridinium Groups for Targeting G‐Quadruplex Structures
2025 C. Platella, S. Di Ciolo, A. Criscuolo, D. Malpicci, R. Gaglione, A. Arciello, D. Musumeci, E. Lucenti, E. Cariati, D. Montesarchio, C. Giannini
Synthesis and Multitarget Inhibitory Effect of Indole-Based Ethyl Cinnamate Derivatives against SARS-CoV-2 Mpro and Cathepsins for Broad-Spectrum Anti-Coronavirus Activity
2025 A. Citarella, G. Sibile, D. Moi, A. Dimasi, T. Braga, L. Dal Col, L. Ruberto, S. Pieraccini, M. Sironi, N. Micale, T. Schirmeister, V. Fasano, A. Silvani, C. Giannini, G. Gribaudo, D. Passarella
Synthesis and multitarget inhibitory effect of indole-based ethyl cinnamate derivatives against SARS-CoV-2 Mpro and cathepsins for broad-spectrum anti-coronavirus activity
2025 A. Citarella, G. Sibille, D. Moi, A. Dimasi, T. Braga, L.D. Col, L. Ruberto, S. Pieraccini, M. Sironi, N. Micale, T. Schirmeister, V. Fasano, A. Silvani, C. Giannini, G. Gribaudo, D. Passarella
Structure-Based Discovery of Hsp90/HDAC6 Dual Inhibitors Targeting Aggressive Prostate Cancer
2025 A. Citarella, S. Belluti, D. Bonanni, D. Moi, I. Piccinini, A. Rinaldi, C. Papulino, R. Benedetti, L. Cuoghi, S.D. Ciolo, A. Silvani, L. Altucci, L. Pinzi, S. Franchini, D. Passarella, C. Sorbi, C. Giannini, C. Imbriano, G. Rastelli
Role of molecular packing in RTP features of positional isomers: The case study of triimidazo-triazine functionalized with ethynyl pyridine moieties
2025 D. Malpicci, S. Di Ciolo, E. Cariati, E. Lucenti, D. Marinotto, D. Maver, C. Giannini, L. Carlucci, C. Botta, A. Forni
Modular Symmetric Ligands for Selective Recognition of Cancer-Relevant G-Quadruplexes
2024 C. Platella, A. Citarella, M. Manenti, G. Spinelli, R. Gaglione, A. Arciello, C. Riccardi, D. Musumeci, D. Montesarchio, C. Giannini, A. Silvani
Innovative molecular platforms for G-quadruplex stabilization
2024 S. Di Ciolo, B. Airoldi, L.C.M. Pariani, C.F. Morelli, C. Giannini, A. Silvani, D. Malpicci, E. Cariati, E. Lucenti, C. Platella, D. Musumeci, R. Gaglione, A. Arciello, D. Montesarchio
Chemical modifications of aromatic scaffolds for the development of new G4 ligands
2024 S. Di Ciolo, B. Airoldi, L.C.M. Pariani, C.F. Morelli, C. Giannini, A. Silvani, D. Malpicci, E. Cariati, E. Lucenti, C. Platella, D. Musumeci, R. Gaglione, A. Arciello, D. Montesarchio
Innovative molecular platforms for G-quadruplex stabilizatioN
2024 S. Di Ciolo, B. Airoldi, L.C.M. Pariani, C.F. Morelli, C. Giannini, A. Silvani, D. Malpicci, E. Cariati, E. Lucenti, C. Platella, D. Musumeci, R. Gaglione, A. Arciello, D. Montesarchio
Synthesis of α-fluorocinnamate derivatives as novel cathepsin S inhibitors with in vitro antiproliferative activity against pancreatic cancer cells
2024 A. Citarella, S. Petrella, D. Moi, A. Dimasi, T. Braga, L. Ruberto, S. Pieraccini, M. Sironi, N. Micale, T. Schirmeister, G. Damia, V. Fasano, A. Silvani, C. Giannini, D. Passarella
Discovery of a Novel Trifluoromethyl Diazirine Inhibitor of SARS-CoV-2 Mpro
2023 A. Citarella, D. Moi, M. Pedrini, H. Pérez-Peña, S. Pieraccini, C. Stagno, N. Micale, T. Schirmeister, G. Sibille, G. Gribaudo, A. Silvani, D. Passarella, C. Giannini
Stimuli responsive features of organic RTP materials: an intriguing carbazole‐cyclic triimidazole derivative
2023 D. Malpicci, A. Forni, C. Botta, C. Giannini, E. Lucenti, D. Marinotto, D. Maver, L. Carlucci, E.M. Cariati
Dual fluorescence and RTP features of carbazole-cyclic triimidazole derivatives: The fluorophores’ connectivity does matter
2023 D. Malpicci, A. Forni, C. Botta, C. Giannini, E. Lucenti, D. Marinotto, D. Maver, L. Carlucci, E. Cariati
Synthesis of SARS-CoV-2 Mpro Inhibitors bearing a Cinnamic Ester Warhead with In Vitro Activity against Human Coronaviruses
2023 A. Citarella, D. Moi, M. Pedrini, H. Pérez-Peña, S. Pieraccini, A. Dimasi, C. Stagno, N. Micale, T. Schirmeister, G. Sibille, G. Gribaudo, A. Silvani, C. Giannini, D. Passarella
Novel Small Multilamellar Liposomes Containing Large Quantities of Peptide Nucleic Acid Selectively Kill Breast Cancer Cells
2022 G. Proshkina, E. Shramova, A. Ryabova, L. Katrivas, C. Giannini, D. Malpicci, Y. Levi-Kalisman, S. Deyev, A. Kotlyar
Aminotriazoloquinazoline- and Aminotriazolo-based Hydroxamic Acids are Novel Potent and Selective HDAC6 Inhibitors with Subnanomolar Activity
2022 A. Citarella, D. Moi, D. Bonanni, L. Pinzi, S. DI CIOLO, D. Passarella, A. Silvani, C. Giannini, G. Rastelli
Synthesis of potent and selective HDAC6 inhibitors led to unexpected opening of a quinazoline ring
2022 D. Moi, A. Citarella, D. Bonanni, L. Pinzi, D. Passarella, A. Silvani, C. Giannini, G. Rastelli
Pyrene-substituted cyclic triimidazole: An appealing and versatile luminescent scaffold for explosive detection
2022 M. Formenti, D. Blasi, E. Cariati, L. Carlucci, A. Forni, C. Giannini, M. Guidotti, S. Econdi, D. Malpicci, D. Marinotto, E. Lucenti
Cyclic Triimidazoles as Stabilizers for Gene Promoter and Human Telomeric DNA G‐Quadruplexes
2022 D. Malpicci, S. Andolina, S. Di Ciolo, E. Lucenti, E. Cariati, S. Marzano, B. Pagano, J. Amato, A. Randazzo, C. Giannini
Room temperature phosphorescence from organic materials: unravelling the emissive behaviour of chloro‐substituted derivatives of cyclic triimidazole
2021 C. Giannini, A. Forni, D. Malpicci, E. Lucenti, D. Marinotto, A. Previtali, L. Carlucci, E. Cariati