CITARELLA, ANDREA
CITARELLA, ANDREA
Dipartimento di Chimica
PROTAC-mediated degradation of peroxisomal d-aspartate oxidase: A novel strategy to modulate d-aspartate homeostasis for schizophrenia treatment
2026 M. Galli, V. Rabattoni, M. Cavinato, F. Vasile, I. Gado, K. Ulfat, H. Shehi, A. Silvani, D. Passarella, A. Citarella, L. Pollegioni, M. Nardini
Stereodefined synthesis of 3-difluoromethyl-benzoxaboroles: novel antimicrobials with unlocked H-bonding
2026 A. Dimasi, A. Montoli, C. Lutti, A. Citarella, P. Ronchi, F. Castagnini, V. Mileo, G. Macetti, V. Baldelli, E. Rossi, P. Landini, D. Passarella, V. Fasano
Design, synthesis and biological evaluation of PROTACs targeting hDASPO
2025 M. Galli, A. Citarella, M. Cavinato, I. Gado, V. Rabattoni, H. Shehi, M. Nardini, A. Silvani, V. Fasano, F. Vasile, L. Pollegioni, D. Passarella
Synthesis and multitarget inhibitory effect of indole-based ethyl cinnamate derivatives against SARS-CoV-2 Mpro and cathepsins for broad-spectrum anti-coronavirus activity
2025 A. Citarella, G. Sibille, D. Moi, A. Dimasi, T. Braga, L.D. Col, L. Ruberto, S. Pieraccini, M. Sironi, N. Micale, T. Schirmeister, V. Fasano, A. Silvani, C. Giannini, G. Gribaudo, D. Passarella
Structure-Based Discovery of Hsp90/HDAC6 Dual Inhibitors Targeting Aggressive Prostate Cancer
2025 A. Citarella, S. Belluti, D. Bonanni, D. Moi, I. Piccinini, A. Rinaldi, C. Papulino, R. Benedetti, L. Cuoghi, S.D. Ciolo, A. Silvani, L. Altucci, L. Pinzi, S. Franchini, D. Passarella, C. Sorbi, C. Giannini, C. Imbriano, G. Rastelli
Mechanistic insights into the base-mediated deuteration of pyridyl phosphonium and ammonium salts
2025 A. Montoli, A. Dimasi, M. Guarnaccia, A. Citarella, P. Ronchi, D. Blasi, S. Rossi, D. Passarella, V. Fasano
Design, synthesis and in vitro validation of bivalent binders of SARS-CoV-2 spike protein: Obeticholic, betulinic and glycyrrhetinic acids as building blocks
2025 M. Pedrini, L. Pozzi, F. Sacchi, A. Citarella, V. Fasano, P. Seneci, S. Pieraccini, L. Ruberto, H. Perez Peña, A. Garzino-Demo, A. Vitiello, L. Sernicola, A. Borsetti, A. Calistri, C. Parolin, D. Passarella
Asymmetric Total Synthesis of (−)‐Glycybridin B, a Pharmacophore Screened Candidate for Tubulin Binding
2025 A. Maiocchi, M. Shevelev, Z. Boiarska, J. Estévez‐gallego, F. Bonato, P. Orlando, A. Chinosi, E. Marcone, A. Citarella, D. Horvath, M.O. Steinmetz, A.E. Prota, A. Varnek, V. Fasano, D. Passarella
Cannabizetol, a Novel Cannabinoid: Chemical Synthesis, Anti-inflammatory Activity and Extraction from Cannabis sativa L
2025 L. Pozzi, A. Gotti, M. Fumagalli, A. Citarella, V. Fasano, G. Paladino, U. Ciriello, S. Princiotto, F. Annunziata, G. Martinelli, E. Sangiovanni, A. Pinto, M. Dell’Agli, D. Passarella
Functionalization of E3 ligase recruiters in the green solvent Cyrene: a sustainable approach for the synthesis of PROTACs precursors
2025 M. Galli, A. Citarella, A. Silvani
Functionalization of E3-ligase recruiters in the green solvent Cyrene: a sustainable approach for the synthesis of PROTAC precursors
2025 M. Galli, A. Citarella, A. Silvani
PROTAC technology for the degradation of hDASPO: from design to synthesis to biophysical and cellular evaluation
2025 M. Galli, A. Citarella, M. Cavinato, I. Gado, V. Rabattoni, H. Shehi, M. Nardini, A. Silvani, V. Fasano, F. Vasile, L. Pollegioni, D. Passarella
Sustainable Synthesis of 1,2,3‐Triazoles using Cyrene as a Biodegradable Solvent in Click Chemistry
2025 A. Citarella, A. Fiori, A. Silvani, D. Passarella, V. Fasano
Synthesis and Multitarget Inhibitory Effect of Indole-Based Ethyl Cinnamate Derivatives against SARS-CoV-2 Mpro and Cathepsins for Broad-Spectrum Anti-Coronavirus Activity
2025 A. Citarella, G. Sibile, D. Moi, A. Dimasi, T. Braga, L. Dal Col, L. Ruberto, S. Pieraccini, M. Sironi, N. Micale, T. Schirmeister, V. Fasano, A. Silvani, C. Giannini, G. Gribaudo, D. Passarella
Self-Assembled Cannabigerol-Based Nanoparticles: Design, Synthesis, and Antiproliferative Activity
2025 A. Amenta, G. Nordio, F. Piazzola, M.L. Di Paolo, F. Milani, M. Giacomini, A. Citarella, U. Ciriello, G. Paladino, S. Pellegrino, F. Silvestri, V. Fasano, L. Dalla Via, D. Passarella
Metal‐Free, Selective Ortho‐Deuteration of N‐Heterocyclic Oxides
2025 A. Montoli, A. Dimasi, A. Citarella, P. Ronchi, D. Passarella, V. Fasano
Revisiting the Reduction of Vinpocetine
2025 S. Borsoi, L. Pozzi, V. Fasano, A. Citarella, G. Macetti, L.L. Presti, G. Paladino, U. Ciriello, D. Passarella
Rotational Motion in Bispidines: A Conformational Study
2025 F. Migliano, L. Pozzi, A. Citarella, G. Macetti, L. Lo Presti, D. Passarella, V. Fasano
Nirmatrelvir: from discovery to modern and alternative synthetic approaches
2024 M. Galli, F. Migliano, V. Fasano, A. Silvani, D. Passarella, A. Citarella
Synthesis of α-fluorocinnamate derivatives as novel cathepsin S inhibitors with in vitro antiproliferative activity against pancreatic cancer cells
2024 A. Citarella, S. Petrella, D. Moi, A. Dimasi, T. Braga, L. Ruberto, S. Pieraccini, M. Sironi, N. Micale, T. Schirmeister, G. Damia, V. Fasano, A. Silvani, C. Giannini, D. Passarella