CITARELLA, ANDREA
CITARELLA, ANDREA
Dipartimento di Chimica
Syntheses, reactivity, and biological applications of coumarins
2024 A. Citarella, S. Vittorio, C. Dank, L. Ielo
PCSK9 inhibitors: a patent review 2018-2023
2024 E.M.A. Fassi, A. Citarella, M. Albani, E.G. Milano, L. Legnani, C. Lammi, A. Silvani, G. Grazioso
First Total Synthesis of Caerulomycin K: A Case Study on Selective, Multiple C-H Functionalizations of Pyridines
2024 A. Dimasi, M. Failla, A. Montoli, A. Citarella, P. Ronchi, D. Passarella, V. Fasano
A Green Approach to Nucleophilic Aromatic Substitutions of Nicotinic Esters in Cyrene
2024 A. Citarella, M. Cavinato, A. Amenta, M. Nardini, A. Silvani, D. Passarella, V. Fasano
Modular Symmetric Ligands for Selective Recognition of Cancer-Relevant G-Quadruplexes
2024 C. Platella, A. Citarella, M. Manenti, G. Spinelli, R. Gaglione, A. Arciello, C. Riccardi, D. Musumeci, D. Montesarchio, C. Giannini, A. Silvani
Recent Advances in SARS-CoV-2 Main Protease Inhibitors: From Nirmatrelvir to Future Perspectives
2023 A. Citarella, A. Dimasi, D. Moi, D. Passarella, A. Scala, A. Piperno, N. Micale
Discovery of potent pyrrolo-pyrimidine and purine HDAC inhibitors for the treatment of advanced prostate cancer
2023 D. Moi, D. Bonanni, S. Belluti, P. Linciano, A. Citarella, S. Franchini, C. Sorbi, C. Imbriano, L. Pinzi, G. Rastelli
Synthesis of SARS-CoV-2 Mpro Inhibitors bearing a Cinnamic Ester Warhead with In Vitro Activity against Human Coronaviruses
2023 A. Citarella, D. Moi, M. Pedrini, H. Pérez-Peña, S. Pieraccini, A. Dimasi, C. Stagno, N. Micale, T. Schirmeister, G. Sibille, G. Gribaudo, A. Silvani, C. Giannini, D. Passarella
Selective noncovalent proteasome inhibiting activity of trifluoromethyl-containing gem-quaternary aziridines
2023 L. Ielo, V. Patamia, A. Citarella, T. Schirmeister, C. Stagno, A. Rescifina, N. Micale, V. Pace
Discovery of a Novel Trifluoromethyl Diazirine Inhibitor of SARS-CoV-2 Mpro
2023 A. Citarella, D. Moi, M. Pedrini, H. Pérez-Peña, S. Pieraccini, C. Stagno, N. Micale, T. Schirmeister, G. Sibille, G. Gribaudo, A. Silvani, D. Passarella, C. Giannini
Computational Design, Synthesis, and Biophysical Evaluation of β-Amido Boronic Acids as SARS-CoV-2 Mpro Inhibitors
2023 E.M.A. Fassi, M. Manenti, A. Citarella, M. Dei Cas, S. Casati, N. Micale, T. Schirmeister, G. Roda, A. Silvani, G. Grazioso
Synthesis of potent and selective HDAC6 inhibitors led to unexpected opening of a quinazoline ring
2022 D. Moi, A. Citarella, D. Bonanni, L. Pinzi, D. Passarella, A. Silvani, C. Giannini, G. Rastelli
Aminotriazoloquinazoline- and Aminotriazolo-based Hydroxamic Acids are Novel Potent and Selective HDAC6 Inhibitors with Subnanomolar Activity
2022 A. Citarella, D. Moi, D. Bonanni, L. Pinzi, S. DI CIOLO, D. Passarella, A. Silvani, C. Giannini, G. Rastelli
Novel Class of Proteasome Inhibitors: In Silico and In Vitro Evaluation of Diverse Chloro(trifluoromethyl)aziridines
2022 L. Ielo, V. Patamia, A. Citarella, T. Efferth, N. Shahhamzehei, T. Schirmeister, C. Stagno, T. Langer, A. Rescifina, N. Micale, V. Pace
Cyrene: A Green Solvent for the Synthesis of Bioactive Molecules and Functional Biomaterials
2022 A. Citarella, A. Amenta, D. Passarella, N. Micale
Synthesis, computational investigation and biological evaluation of α,α-difluoromethyl ketones embodying pyrazole and isoxazole nuclei as COX inhibitors
2022 A. Citarella, L. Ielo, C. Stagno, M. Cristani, C. Muscara, V. Pace, N. Micale
Dual Targeting Strategies on Histone Deacetylase 6 (HDAC6) and Heat Shock Protein 90 (Hsp90)
2022 D. Bonanni, A. Citarella, D. Moi, L. Pinzi, E. Bergamini, G. Rastelli
Hydroxamic Acid Derivatives: From Synthetic Strategies to Medicinal Chemistry Applications
2021 A. Citarella, D. Moi, L. Pinzi, D. Bonanni, G. Rastelli
Natural product-based hybrids as potential candidates for the treatment of cancer: Focus on curcumin and resveratrol
2021 N. Micale, M.S. Molonia, A. Citarella, F. Cimino, A. Saija, M. Cristani, A. Speciale
Pseudo-dipeptide bearing α,α-difluoromethyl ketone moiety as electrophilic warhead with activity against coronaviruses
2021 A. Citarella, D. Gentile, A. Rescifina, A. Piperno, B. Mognetti, G. Gribaudo, M.T. Sciortino, W. Holzer, V. Pace, N. Micale