GRAZIOSO, GIOVANNI

GRAZIOSO, GIOVANNI  

Dipartimento di Scienze Farmaceutiche  

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Titolo Data di pubblicazione Autori Tipo File Abstract
Ago-allosteric modulation of nicotinic alpha7 receptors : a mechanistic insight by metadynamics and essential dynamics 11-giu-2014 G. Grazioso Conference Object -
Agonisti nicotinici selettivi nel trattamento di patologie del Sistema Nervoso Centrale 16-set-2007 C. De MicheliM. De AmiciC. DallanoceG. GraziosoL. RizziP. MagroneC. Matera Book Part (author) -
Alkene Epoxidations Mediated by Mn-Salen Macrocyclic Catalysts 2-apr-2021 G. Grazioso + Article (author) -
Allosteric modulation of alpha7 nicotinic receptors : mechanistic insight through metadynamics and essential dynamics 28-dic-2015 G. GraziosoC. MateraC. DallanoceM. De Amici + Article (author) -
Alpha7 nicotinic acetylcholine receptor agonists: prediction of their binding affinity through a molecular mechanics poisson-boltzmann surface area approach 1-gen-2008 G. GraziosoM. De AmiciC. De Micheli + Article (author) -
Analytical, computational and formulation studies on TPGS as P-gp inhibitor 1-nov-2015 M.D.Del CurtoC. BolchiA. FoppoliL. FumagalliF. SelminG. GraziosoL. Palugan Book Part (author) -
Application of the Ugi reaction with multiple amino acid-derived components : synthesis and conformational evaluation of piperazine-based minimalist peptidomimetics 22-apr-2015 M. StucchiM. ChristodoulouG. GraziosoA. SilvaniG. Lesma + Article (author) -
Bifunctional compounds targeting both D2 and non-α7 nACh receptors: design, synthesis and pharmacological characterization 28-ago-2015 C. MateraL. PucciG. GraziosoF. ClementiM. De AmiciC. Dallanoce + Article (author) -
Bioactive cyclization optimizes the affinity of a proprotein convertase subtilisin/kexin type 9 (PCSK9) peptide inhibitor 11-mar-2021 Lammi C.Grazioso G. + Article (author) -
Biological Characterization of Computationally Designed Analogs of peptide TVFTSWEEYLDWV (Pep2-8) with Increased PCSK9 Antagonistic Activity 20-feb-2019 C. LammiA. ArnoldiG. Grazioso + Article (author) -
Computational approaches in the rational design of improved carbonyl quenchers : focus on histidine containing dipeptides 1-set-2016 G. VistoliM. ColzaniA. MazzolariG. GraziosoA. PedrettiM. CariniG. Aldini + Article (author) -
Computational Design and Biological Evaluation of Analogs of Lupin Peptide P5 Endowed with Dual PCSK9/HMG-CoAR Inhibiting Activity 18-mar-2022 C. LammiE. FassiJ. LiM. BartolomeiG. RodaA. ArnoldiG. Grazioso + Article (author) -
COMPUTATIONAL INVESTIGATION ON SUBSTRATE UPTAKE AND RELEASE IN A GLUTAMATE TRANSPORTER 17-apr-2012 G. GraziosoC. De Micheli + Conference Object -
Computationally Driven Structure Optimization, Synthesis, and Biological Evaluation of Imidazole-Based Proprotein Convertase Subtilisin/Kexin 9 (PCSK9) Inhibitors 18-giu-2019 Lammi, CarmenArnoldi, AnnaLesma, GiordanoSilvani, AlessandraGrazioso, Giovanni + Article (author) -
Covalent docking of selected boron-based serine beta-lactamase inhibitors 1-mag-2015 G. Grazioso + Article (author) -
Design and synthesis of selective ligands targeting different nAChR subtypes 27-feb-2014 M. QuadriC. MateraG. GraziosoM. De AmiciC. Dallanoce Conference Object -
Design of Cyclopentaisoxazoline Amino Acids as Conformationally Constrained Agonists at Glutamate Receptors 3-nov-2003 P. ContiM. De AmiciG. GraziosoG. RodaC. De Micheli + Article (author) -
Design of novel α7-subtype-preferring nicotinic acetylcholine receptor agonists: application of docking and MM-PBSA computational approaches, synthetic and pharmacological studies 1-gen-2009 G. GraziosoC. MateraF. FrigerioL. PucciC. DallanoceM. De Amici + Article (author) -
DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF PEPTIDOMIMETIC FALCIPAIN-2 INHIBITORS AS ANTIMALARIAL AGENTS 17-apr-2012 G. Grazioso + Conference Object -
Design, Synthesis, and Pharmacological Characterization of Novel Spirocyclic Quinuclidinyl-Δ2-Isoxazoline Derivatives as Potent and Selective Agonists of α7 Nicotinic Acetylcholine Receptors 2-mag-2011 C.M.L. DallanoceP. MagroneC. MateraF. FrigerioG. GraziosoM. DE AMICIL. PucciF. ClementiC. DE MICHELI + Article (author) -