CAZZANIGA, GIULIA
CAZZANIGA, GIULIA
Dipartimento di Scienze Farmaceutiche
5-(4-Nitrophenyl)furan-2-carboxylic Acid
2022 M. Mori, A. Tresoldi, S. Villa, G. Cazzaniga, M. Bellinzoni, F. Meneghetti
6-Hydroxy-2-methylbenzofuran-4-carboxylic acid
2020 M. Mori, F. Meneghetti, L.R. Chiarelli, A. Diego, D. Nava, A. Gelain, G. Cazzaniga, S. Villa, E.R.E. Pini
A dual-target approach in anti-tuberculosis therapy: new MptpB/MbtI inhibitors
2020 G. Cazzaniga, M. Mori, A. Gelain, E. Pini, G. Stelitano, L.R. Chiarelli, F. Meneghetti, S. Villa
Biological Screening and Crystallographic Studies of Hydroxy γ-Lactone Derivatives to Investigate PPARγ Phosphorylation Inhibition
2023 D. Capelli, G. Cazzaniga, M. Mori, A. Laghezza, F. Loiodice, M. Quaglia, E. Negro, F. Meneghetti, S. Villa, R. Montanari
Development of a novel approach to overcome biofilm formation by natural product derivatives
2022 A. Gelain, G. Cazzaniga, M. Mori, P.J. Molino, P. Hajes, F. Villa, C. Cattò, F. Cappitelli, S. Villa
Insights on the Modulation of SIRT5 Activity: A Challenging Balance
2022 M. Mori, G. Cazzaniga, F. Meneghetti, S. Villa, A. Gelain
Low-Molecular-Weight Phosphatase B (LMW-MPtpB) inhibition as a strategy to identify new drug candidates against tuberculosis
2021 M. Mori, G. Cazzaniga, L.R. Chiarelli, G. Stelitano, S. Ciceri, T. Tuccinardi, G. Poli, F. Meneghetti, S. Villa
Methyl 5-(2-Fluoro-4-nitrophenyl)furan-2-carboxylate
2022 M. Mori, A. Tresoldi, G. Cazzaniga, F. Meneghetti, S. Villa
Native llama Nanobody Library Panning Performed by Phage and Yeast Display Provides Binders Suitable for C-Reactive Protein Detection
2021 S. Oloketuyi, R. Bernedo, A. Christmann, J. Borkowska, G. Cazzaniga, H.W. Schuchmann, J. Niedziółka-Jönsson, K. Szot-Karpińska, H. Kolmar, A. de Marco
Natural products against key Mycobacterium tuberculosis enzymatic targets : Emerging opportunities for drug discovery
2021 G. Cazzaniga, M. Mori, L. Roberto Chiarelli, A. Gelain, F. Meneghetti, S. Villa
New strategies to overcome biofilm formation by natural product derivatives
2022 S. Villa, G. Cazzaniga, M. Mori, P.J. Molino, P. Hayes, F. Villa, C. Cattò, F. Cappitelli, A. Gelain
Phagocyte-targeting polymersomes as intracellular delivery carriers for enzymatic inhibitors with antitubercular activity
2022 G. Cazzaniga, M. Mori, F. Meneghetti, L.R. Chiarelli, G. Stelitano, C. Di Gugliemo, I.L. Batalha, G. Battaglia, S. Villa
Polymersomes as selective drug delivery carriers for innovative anti-TB agents
2022 G. Cazzaniga, M. Mori, F. Meneghetti, L.R. Chiarelli, G. Stelitano, I.L. Batalha, G. Battaglia, S. Villa
Synthesis and Assessment of the In Vitro and Ex Vivo Activity of Salicylate Synthase (Mbti) Inhibitors as New Candidates for the Treatment of Mycobacterial Infections
2022 M. Mori, G. Stelitano, A. Griego, L.R. Chiarelli, G. Cazzaniga, A. Gelain, E. Pini, M. Camera, P. Canzano, A. Fumagalli, E. Scarpa, C. Cordiglieri, L. Rizzello, S. Villa, F. Meneghetti
Synthesis, Characterization, and Biological Evaluation of New Derivatives Targeting MbtI as Antitubercular Agents
2021 M. Mori, G. Stelitano, L.R. Chiarelli, G. Cazzaniga, A. Gelain, D. Barlocco, E.R.E. Pini, F. Meneghetti, S. Villa
Targeting Siderophore-Mediated Iron Uptake in M. abscessus: A New Strategy to Limit the Virulence of Non-Tuberculous Mycobacteria
2023 M. Mori, G. Stelitano, G. Cazzaniga, A. Gelain, A. Tresoldi, M. Cocorullo, M. Roversi, L.R. Chiarelli, M. Tomaiuolo, P. Delre, G. Felice Mangiatordi, A. Griego, L. Rizzello, A. Cassetta, S. Covaceuszach, S. Villa, F. Meneghetti
Targeting the mycobactin biosynthesis pathway in M. tuberculosis: a step towards the improvement of the anti-virulence activity of MbtI inhibitors
2022 M. Mori, S. Villa, L.R. Chiarelli, G. Stelitano, A. Gelain, G. Cazzaniga, M. Bellinzoni, L. Rizzello, E. Scarpa, A. Griego, A. Fumagalli, F. Meneghetti
Unraveling the interaction mechanism of a benzothiadiazole-2.2-dioxide derivative with STAT3 : towards novel direct inhibitors
2021 M. Mori, E. Gilardoni, L. Regazzoni, A. Pedretti, D. Colombo, G. Parkinson, A. Asai, G. Cazzaniga, F. Meneghetti, S. Villa, A. Gelain
Virtual screening and crystallographic studies reveal an unexpected γ-lactone derivative active against MptpB as a potential antitubercular agent
2022 G. Cazzaniga, M. Mori, F. Meneghetti, L.R. Chiarelli, G. Stelitano, I. Caligiuri, F. Rizzolio, S. Ciceri, G. Poli, D. Staver, G. Ortore, T. Tuccinardi, S. Villa
γ-hidroxy-lactone derivatives as ppar-γ non-agonists blocking cdk5-mediated phosporylation for a safer anti-diabetic treatment
2023 G. Cazzaniga, M. Mori, D. Capelli, R. Montanari, A. Laghezza, F. Loiodice, I. Bassanini, S. Romeo, E.M.A. Fassi, M. Quaglia, G. Grazioso, F. Meneghetti, S. Villa