BORSARI, CHIARA
BORSARI, CHIARA
Dipartimento di Scienze Farmaceutiche
From Batch to Flow: Chemo-Enzymatic Asymmetric Synthesis of Piperidine Scaffolds
2025 S. Vicinanza, S. Patti, M. Pirotta, I. Magrini Alunno, F. Annunziata, R. Gandolfi, C. Borsari, I. Bassanini, D. Monti, E. Elisa Ferrandi, L. Tamborini
Chemo-enzymatic asymmetric flow synthesis of piperidine as pharmaceutically relevant scaffolds
2025 S. Vicinanza, S. Patti, M. Pirotta, I. Magrini Alumno, F. Annunziata, R. Gandolfi, C. Borsari, I. Bassanini, D. Monti, E. Elisa Ferrandi, L. Tamborini
The European Federation for Medicinal Chemistry and Chemical Biology (EFMC) Best Practice Initiative: Hit to Lead
2025 J. Quancard, A. Bach, C. Borsari, R. Craft, C. Gnamm, S.M. Guéret, I.V. Hartung, H.F. Koolman, S. Laufer, S. Lepri, J. Messinger, K. Ritter, G. Sbardella, A. Unzue Lopez, M.K. Willwacher, B. Cox, R.J. Young
Highlights from the Lowlands: Early Career Researchers Shine at Medicinal Chemistry Frontiers 2024
2025 S.M. Mckenna, C. Borsari, S. Chin Chan, E.J. Donckele, F.F. Faucher, M.C. Grenier‐davies, K. Haranahalli, B. Matagne, A. Monastyrskyi, R. Petracca
Two-Step Flow Amidation of Natural Phenolic Acids as Antiradical and Antimicrobial Agents
2025 D. Pecora, A.M. Magni, S. Vicinanza, F. Annunziata, S. Princiotto, S. Donzella, G. Meroni, P.A. Martino, N. Basilico, S. Parapini, P. Conti, C. Borsari, L. Tamborini
From pan-active to parasite-selective antiparasitic agents: A scaffold hopping approach
2025 C. Borsari, N. Santarem, D. Coertzen, A. Mazzolari, A.I. Corfu, C. Coelho, F. Barbosa, L. Tamborini, L.-. Birkholtz, L. Raffellini, O. Keminer, N. Basilico, S. Parapini, S. Gul, A. Cordeiro-da-Silva, P. Conti
Tyrosol and hydroxytyrosol carbonates and carbamates as novel antiradical and antimicrobial agents: a chemo-enzymatic flow synthesis
2024 S. Vicinanza, L. Mombelli, F. Annunziata, S. Donzella, M.L. Contente, C. Borsari, G. Meroni, P.A.M. Martino, A. Pinto, L. Tamborini
TRIAZINE DERIVATIVE AS COVALENT INHIBITORS OF PI3K | [TRIAZINDERIVAT ALS KOVALENTE INHIBITOREN VON PI3K]
2024 M. Wymann, C. Borsari
Targeted Covalent Inhibitors in Drug Discovery, Chemical Biology and Beyond
2024 R.A.M. Serafim, M. Gehringer, C. Borsari
METHOD FOR IDENTIFYING PI3 KINASE-ALPHA INHIBITORS
2024 C. Borsari, M. Wymann
TRIAZINE DERIVATIVE AS COVALENT INHIBITORS OF PI3K
2024 M. Wymann, C. Borsari
A high affinity pan-PI3K binding module supports selective targeted protein degradation of PI3Kα
2024 W.T. Jauslin, M. Schild, T. Schaefer, C. Borsari, C. Orbegozo, L. Bissegger, S. Zhanybekova, D. Ritz, A. Schmidt, M. Wymann, D. Gillingham
Chemo-enzymatic flow synthesis of nature-inspired phenolic carbonates and carbamates as antimicrobial and antiradical agents
2024 F. Annunziata, S. Vicinanza, L. Mombelli, S. Donzella, G. Meroni, C. Borsari, M.L. Contente, P.A. Martino, P. Conti, A. Pinto, S. Dallavalle, L. Tamborini
Rapid, potent, and persistent covalent chemical probes to deconvolute PI3Kα signaling
2024 L. Bissegger, T.A. Constantin, E. Keles, L. Raguž, I. Barlow-Busch, C. Orbegozo, T. Schaefer, V. Borlandelli, T. Bohnacker, R. Sriramaratnam, A. Schäfer, M. Gstaiger, J.E. Burke, C. Borsari, M.P. Wymann
TRIAZINE DERIVATIVE AS REVERSIBLE AND IRREVERSIBLE COVALENT INHIBITORS OF PI3K | [TRIAZINDERIVAT ALS REVERSIBLE UND IRREVERSIBLE KOVALENTE PI3K-HEMMER]
2024 C. Borsari, M. Wymann
METHOD FOR IDENTIFYING PI3 KINASE-ALPHA INHIBITORS | [VERFAHREN ZUR IDENTIFIZIERUNG VON PI3-KINASE-ALPHA-INHIBITOREN]
2024 C. Borsari, M. Wymann
TRIAZINE DERIVATIVE AS REVERSIBLE AND IRREVERSIBLE COVALENT INHIBITORS OF PI3K
2024 C. Borsari, M. Wymann
Chemo-enzymatic flow synthesis of nature-inspired phenolic carbonates and carbamates as antiradical and antimicrobial agents
2024 S. Vicinanza, L. Mombelli, F. Annunziata, S. Donzella, M.L. Contente, C. Borsari, P. Conti, G. Meroni, F. Molinari, P.A.M. Martino, A. Pinto, L. Tamborini
Boosting the Impact of EFMC Young Scientists Network Through the Creation of Working Groups
2024 M. Mari, C. Lanthier, M. Proj, E.J. Donckele, L. Josa‐culleré, K. Goncharenko, S. Leroy, B. Matagne, S.M. Mckenna, C. Borsari
Discovery of 1,3,4-Oxadiazole Derivatives as Broad-Spectrum Antiparasitic Agents
2024 A.I. Corfu, N. Santarem, S. Luelmo, G. Mazza, A. Greco, A. Altomare, G. Ferrario, G. Nasta, O. Keminer, G. Aldini, L. Tamborini, N. Basilico, S. Parapini, S. Gul, A. Cordeiro-da-Silva, P. Conti, C. Borsari