BORSARI, CHIARA
BORSARI, CHIARA
Dipartimento di Scienze Farmaceutiche
Chemo-enzymatic flow synthesis of chiral piperidine scaffolds
2026 S. Vicinanza, S. Patti, M. Pirotta, I. Magrini Alunno, F. Annunziata, R. Gandolfi, C. Borsari, I. Bassanini, D. Monti, E. Elisa Ferrandi, L. Tamborini
Fifteen Years, One Mission: Innovative, Inspirational, and Impactful Discoveries
2026 S.V. Bigi-Botterill, C. Borsari, A.W. Dombrowski, M.A. Estrada, M.P. Farrell, A.P. Riley, J.G. Woodland
Development of First-in-Class Covalent Inhibitors of PFKFB3 for PDAC treatment
2025 G. Antonini, A. Fiore, A. Scarano, A.I. Corfu, L. Sicuro, R. Pacchiana, M. Donadelli, L. Mollica, L. Tamborini, P. Conti, S. Bruno, C. Borsari
Highlights from the Lowlands: Early Career Researchers Shine at Medicinal Chemistry Frontiers 2024
2025 S.M. Mckenna, C. Borsari, S. Chin Chan, E.J. Donckele, F.F. Faucher, M.C. Grenier‐davies, K. Haranahalli, B. Matagne, A. Monastyrskyi, R. Petracca
Two-Step Flow Amidation of Natural Phenolic Acids as Antiradical and Antimicrobial Agents
2025 D. Pecora, A.M. Magni, S. Vicinanza, F. Annunziata, S. Princiotto, S. Donzella, G. Meroni, P.A. Martino, N. Basilico, S. Parapini, P. Conti, C. Borsari, L. Tamborini
In This Issue
2025 C. Borsari
From Batch to Flow: Chemo-Enzymatic Asymmetric Synthesis of Piperidine Scaffolds
2025 S. Vicinanza, S. Patti, M. Pirotta, I. Magrini Alunno, F. Annunziata, R. Gandolfi, C. Borsari, I. Bassanini, D. Monti, E. Elisa Ferrandi, L. Tamborini
The European Federation for Medicinal Chemistry and Chemical Biology (EFMC) Best Practice Initiative: Hit to Lead
2025 J. Quancard, A. Bach, C. Borsari, R. Craft, C. Gnamm, S.M. Guéret, I.V. Hartung, H.F. Koolman, S. Laufer, S. Lepri, J. Messinger, K. Ritter, G. Sbardella, A. Unzue Lopez, M.K. Willwacher, B. Cox, R.J. Young
From pan-active to parasite-selective antiparasitic agents: A scaffold hopping approach
2025 C. Borsari, N. Santarem, D. Coertzen, A. Mazzolari, A.I. Corfu, C. Coelho, F. Barbosa, L. Tamborini, L.-. Birkholtz, L. Raffellini, O. Keminer, N. Basilico, S. Parapini, S. Gul, A. Cordeiro-da-Silva, P. Conti
Announcing the Early Career Board of Journal of Medicinal Chemistry
2025 M. Ashley, C. Borsari, S. Cazzamalli, J. Chu, Y. Lee, P. Perlíková, R.C. Sarott, B.J. Simmons, X. Xu, N.A. Patil, C. Kounde, S. Wang
Chemo-enzymatic asymmetric flow synthesis of piperidine as pharmaceutically relevant scaffolds
2025 S. Vicinanza, S. Patti, M. Pirotta, I. Magrini Alumno, F. Annunziata, R. Gandolfi, C. Borsari, I. Bassanini, D. Monti, E. Elisa Ferrandi, L. Tamborini
Tyrosol and hydroxytyrosol carbonates and carbamates as novel antiradical and antimicrobial agents: a chemo-enzymatic flow synthesis
2024 S. Vicinanza, L. Mombelli, F. Annunziata, S. Donzella, M.L. Contente, C. Borsari, G. Meroni, P.A.M. Martino, A. Pinto, L. Tamborini
TRIAZINE DERIVATIVE AS COVALENT INHIBITORS OF PI3K
2024 M. Wymann, C. Borsari
METHOD FOR IDENTIFYING PI3 KINASE-ALPHA INHIBITORS
2024 C. Borsari, M. Wymann
Targeted Covalent Inhibitors in Drug Discovery, Chemical Biology and Beyond
2024 R.A.M. Serafim, M. Gehringer, C. Borsari
Chemo-enzymatic flow synthesis of nature-inspired phenolic carbonates and carbamates as antimicrobial and antiradical agents
2024 F. Annunziata, S. Vicinanza, L. Mombelli, S. Donzella, G. Meroni, C. Borsari, M.L. Contente, P.A. Martino, P. Conti, A. Pinto, S. Dallavalle, L. Tamborini
Rapid, potent, and persistent covalent chemical probes to deconvolute PI3Kα signaling
2024 L. Bissegger, T.A. Constantin, E. Keles, L. Raguž, I. Barlow-Busch, C. Orbegozo, T. Schaefer, V. Borlandelli, T. Bohnacker, R. Sriramaratnam, A. Schäfer, M. Gstaiger, J.E. Burke, C. Borsari, M.P. Wymann
In This Issue
2024 C. Borsari
Chemo-enzymatic flow synthesis of nature-inspired phenolic carbonates and carbamates as antiradical and antimicrobial agents
2024 S. Vicinanza, L. Mombelli, F. Annunziata, S. Donzella, M.L. Contente, C. Borsari, P. Conti, G. Meroni, F. Molinari, P.A.M. Martino, A. Pinto, L. Tamborini
A high affinity pan-PI3K binding module supports selective targeted protein degradation of PI3Kα
2024 W.T. Jauslin, M. Schild, T. Schaefer, C. Borsari, C. Orbegozo, L. Bissegger, S. Zhanybekova, D. Ritz, A. Schmidt, M. Wymann, D. Gillingham