APPIANI, REBECCA
APPIANI, REBECCA
Dipartimento di Scienze Farmaceutiche
1,4-Benzodioxane, an evergreen, versatile scaffold in medicinal chemistry : a review of its recent applications in drug design
2020 C. Bolchi, F. Bavo, R. Appiani, G. Roda, M. Pallavicini
4-, 5-, 6-, and 7-Hydroxybenzofuran: a unified strategy for a two-step synthesis of versatile benzofuranic building blocks
2022 R. Appiani, C. Morano, G. Roda, M. Pallavicini, C. Bolchi
ALPHA4BETA2 NEURONAL NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS: FROM SUBTYPE SELECTIVE TO STOICHIOMETRIC ISOPHORM SELECTIVE PARTIAL AGONISM.
2023 R. Appiani
Behavioural and pharmacological profiles of zebrafish administrated pyrrolidinyl benzodioxanes and prolinol aryl ethers with high affinity for heteromeric nicotinic acetylcholine receptors
2020 D. Braida, L. Ponzoni, M. Moretti, P. Viani, M. Pallavicini, C. Bolchi, R. Appiani, F. Bavo, C. Gotti, M. Sala
Determinants for α4β2 vs. α3β4 Subtype Selectivity of Pyrrolidine-Based nAChRs Ligands: A Computational Perspective with Focus on Recent cryo-EM Receptor Structures [Determinants for alpha 4 beta 2 vs. alpha 3 beta 4 Subtype Selectivity of Pyrrolidine-Based nAChRs Ligands: A Computational Perspective with Focus on Recent cryo-EM Receptor Structures]
2021 F. Bavo, M. Pallavicini, R. Appiani, C. Bolchi
Efficient conversion of d-mannitol into 1,2:5,6-diacetonide with Aquivion-H as a recyclable catalyst
2021 C. Bolchi, R. Appiani, G. Roda, V. Bertolini, S. Arnoldi, M. Pallavicini
Efficient One-Pot Reductive Aminations of Carbonyl Compounds with Aquivion-Fe as a Recyclable Catalyst and Sodium Borohydride
2020 V. Airoldi, O. Piccolo, G. Roda, R. Appiani, F. Bavo, R. Tassini, S. Paganelli, S. Arnoldi, M. Pallavicini, C. Bolchi
From 2-Triethylammonium Ethyl Ether of 4-Stilbenol (MG624) to Selective Small-Molecule Antagonists of Human α9α10 Nicotinic Receptor by Modifications at the Ammonium Ethyl Residue [From 2-Triethylammonium Ethyl Ether of 4-Stilbenol (MG624) to Selective Small-Molecule Antagonists of Human alpha 9 alpha 10 Nicotinic Receptor by Modifications at the Ammonium Ethyl Residue]
2022 F. Bavo, M. Pallavicini, S. Pucci, R. Appiani, A. Giraudo, B. Eaton, L. Lucero, C. Gotti, M. Moretti, P. Whiteaker, C. Bolchi
Green Oxidation of Ketones to Lactones with Oxone in Water
2021 V. Bertolini, R. Appiani, M. Pallavicini, C. Bolchi
Modifications at C(5) of 2-(2-Pyrrolidinyl)-Substituted 1,4-Benzodioxane Elicit Potent α4β2 Nicotinic Acetylcholine Receptor Partial Agonism with High Selectivity over the α3β4 Subtype
2020 F. Bavo, M. Pallavicini, C. Gotti, R. Appiani, M. Moretti, S.F. Colombo, S. Pucci, P. Viani, R. Budriesi, M. Renzi, S. Fucile, C. Bolchi
Pyrrolidinyl benzofurans and benzodioxanes: Selective α4β2 nicotinic acetylcholine receptor ligands with different activity profiles at the two receptor stoichiometries
2022 R. Appiani, M. Pallavicini, A.K. Hamouda, C. Bolchi
Subnanomolar Affinity and Selective Antagonism at α7 Nicotinic Receptor by Combined Modifications of 2-Triethylammonium Ethyl Ether of 4-Stilbenol (MG624)
2023 F. Bavo, M. Pallavicini, S. Pucci, R. Appiani, A. Giraudo, H. Oh, D.L. Kneisley, B. Eaton, L. Lucero, C. Gotti, F. Clementi, P. Whiteaker, C. Bolchi