GIRAUDO, ALESSANDRO
GIRAUDO, ALESSANDRO
Dipartimento di Scienze Farmaceutiche
Efficient alpha-selective chlorination of phenylacetic acid and its para-substituted analogues†
2025 C. Morano, A. Giraudo, G. Roda, E. Armano, G. Nasta, M. Sipala, M. Pallavicini, C. Bolchi
Identifying Pharmacopoeial Amino Acids through an Instructive Sequence of Physical, Chemical, and Chromatographic Analyses
2025 C. Morano, E. Armano, G. Roda, A. Giraudo, M. Pallavicini, C. Bolchi
Uncovering the Mechanism of Action of Antiprotozoal Agents: A Survey on Photoaffinity Labeling Strategy
2024 A. Giraudo, C. Bolchi, M. Pallavicini, R. Di Santo, R. Costi, F. Saccoliti
Selective potentiation of the (α4)3(β2)2 nicotinic acetylcholine receptor response by NS9283 analogues
2024 R. Appiani, F. Viscarra, P. Biggin, I. Bermudez, A. Giraudo, M. Pallavicini, C. Bolchi
3-Ethoxycarbonyl-1,4-benzodioxin-2-carboxylic Acid
2024 E. Armano, A. Giraudo, C. Morano, M. Pallavicini, C. Bolchi
Subnanomolar Affinity and Selective Antagonism at α7 Nicotinic Receptor by Combined Modifications of 2-Triethylammonium Ethyl Ether of 4-Stilbenol (MG624)
2023 F. Bavo, M. Pallavicini, S. Pucci, R. Appiani, A. Giraudo, H. Oh, D.L. Kneisley, B. Eaton, L. Lucero, C. Gotti, F. Clementi, P. Whiteaker, C. Bolchi
Green Oxidation of Heterocyclic Ketones with Oxone in Water
2023 A. Giraudo, E. Armano, C. Morano, M. Pallavicini, C. Bolchi
Methyl 8- and 5-Nitro-1,4-Benzodioxane-2-Carboxylate
2023 E. Armano, A. Giraudo, C. Morano, M. Pallavicini, C. Bolchi
Methyl 8- and 5-Bromo-1,4-Benzodioxane-2-carboxylate: Unambiguous Identification of the Two Regioisomers
2023 E. Armano, A. Giraudo, M. Pallavicini, C. Bolchi
Small molecule ligands for α9 * and α7 nicotinic receptors: A survey and an update, respectively
2023 A. Giraudo, M. Pallavicini, C. Bolchi
From 2-Triethylammonium Ethyl Ether of 4-Stilbenol (MG624) to Selective Small-Molecule Antagonists of Human α9α10 Nicotinic Receptor by Modifications at the Ammonium Ethyl Residue [From 2-Triethylammonium Ethyl Ether of 4-Stilbenol (MG624) to Selective Small-Molecule Antagonists of Human alpha 9 alpha 10 Nicotinic Receptor by Modifications at the Ammonium Ethyl Residue]
2022 F. Bavo, M. Pallavicini, S. Pucci, R. Appiani, A. Giraudo, B. Eaton, L. Lucero, C. Gotti, M. Moretti, P. Whiteaker, C. Bolchi
Partial rescue of f508del-cftr stability and trafficking defects by double corrector treatment
2021 V. Capurro, V. Tomati, E. Sondo, M. Renda, A. Borrelli, C. Pastorino, D. Guidone, A. Venturini, A. Giraudo, S.M. Bertozzi, I. Musante, F. Bertozzi, T. Bandiera, F. Zara, L.J.V. Galietta, N. Pedemonte
Distinctive lipid signatures of bronchial epithelial cells associated with cystic fibrosis drugs, including Trikafta
2020 N. Liessi, E. Pesce, C. Braccia, S.M. Bertozzi, A. Giraudo, T. Bandiera, N. Pedemonte, A. Armirotti
Five-Membered N-Heterocyclic Scaffolds as Novel Amino Bioisosteres at γ-Aminobutyric Acid (GABA) Type A Receptors and GABA Transporters
2019 A. Giraudo, J. Krall, F. Bavo, B. Nielsen, K.T. Kongstad, B. Rolando, R. De Blasio, D.E. Gloriam, R. Loffler, L. Thiesen, K. Harpsoe, K. Frydenvang, D. Boschi, P. Wellendorph, M.L. Lolli, A.A. Jensen, B. Frolund
Regioselective N-Alkylation of Ethyl 4-Benzyloxy-1,2,3-triazolecarboxylate: A Useful Tool for the Synthesis of Carboxylic Acid Bioisosteres
2019 S. Sainas, A.C. Pippione, A. Giraudo, K. Martina, F. Bosca, B. Rolando, A. Barge, A. Ducime, A. Federico, S.J. Grossert, R.L. White, D. Boschi, M.L. Lolli
Harnessing cavitational effects for green process intensification
2019 Z. Wu, S. Tagliapietra, A. Giraudo, K. Martina, G. Cravotto
Hydroxyazole scaffold-based Plasmodium falciparum dihydroorotate dehydrogenase inhibitors: Synthesis, biological evaluation and X-ray structural studies
2019 A.C. Pippione, S. Sainas, P. Goyal, I. Fritzson, G.C. Cassiano, A. Giraudo, M. Giorgis, T.A. Tavella, R. Bagnati, B. Rolando, R. Caing-Carlsson, F.T.M. Costa, C.H. Andrade, S. Al-Karadaghi, D. Boschi, R. Friemann, M.L. Lolli
4-Hydroxy-1,2,3-triazole moiety as bioisostere of the carboxylic acid function: a novel scaffold to probe the orthosteric γ-aminobutyric acid receptor binding site
2018 A. Giraudo, J. Krall, B. Nielsen, T.E. Sorensen, K.T. Kongstad, B. Rolando, D. Boschi, B. Frolund, M.L. Lolli
Hydroxytriazole derivatives as potent and selective aldo-keto reductase 1C3 (AKR1C3) inhibitors discovered by bioisosteric scaffold hopping approach
2017 A.C. Pippione, A. Giraudo, D. Bonanni, I.M. Carnovale, E. Marini, C. Cena, A. Costale, D. Zonari, K. Pors, M. Sadiq, D. Boschi, S. Oliaro-Bosso, M.L. Lolli