BAVO, FRANCESCO
BAVO, FRANCESCO
Dipartimento di Scienze Farmaceutiche
Subnanomolar Affinity and Selective Antagonism at α7 Nicotinic Receptor by Combined Modifications of 2-Triethylammonium Ethyl Ether of 4-Stilbenol (MG624)
2023 F. Bavo, M. Pallavicini, S. Pucci, R. Appiani, A. Giraudo, H. Oh, D.L. Kneisley, B. Eaton, L. Lucero, C. Gotti, F. Clementi, P. Whiteaker, C. Bolchi
From 2-Triethylammonium Ethyl Ether of 4-Stilbenol (MG624) to Selective Small-Molecule Antagonists of Human α9α10 Nicotinic Receptor by Modifications at the Ammonium Ethyl Residue [From 2-Triethylammonium Ethyl Ether of 4-Stilbenol (MG624) to Selective Small-Molecule Antagonists of Human alpha 9 alpha 10 Nicotinic Receptor by Modifications at the Ammonium Ethyl Residue]
2022 F. Bavo, M. Pallavicini, S. Pucci, R. Appiani, A. Giraudo, B. Eaton, L. Lucero, C. Gotti, M. Moretti, P. Whiteaker, C. Bolchi
Evidence of a dual mechanism of action underlying the anti-proliferative and cytotoxic effects of ammonium-alkyloxy-stilbene-based α7- and α9- nicotinic ligands on glioblastoma cells
2022 S. Pucci, C. Bolchi, F. Bavo, M. Pallavicini, C. De Palma, M. Renzi, S. Fucile, R. Benfante, S. Di Lascio, D. Lattuada, J. Bessereau, M. D'Alessandro, V. Risson, M. Zoli, F. Clementi, C. Gotti
Determinants for α4β2 vs. α3β4 Subtype Selectivity of Pyrrolidine-Based nAChRs Ligands: A Computational Perspective with Focus on Recent cryo-EM Receptor Structures [Determinants for alpha 4 beta 2 vs. alpha 3 beta 4 Subtype Selectivity of Pyrrolidine-Based nAChRs Ligands: A Computational Perspective with Focus on Recent cryo-EM Receptor Structures]
2021 F. Bavo, M. Pallavicini, R. Appiani, C. Bolchi
1,4-Benzodioxane, an evergreen, versatile scaffold in medicinal chemistry : a review of its recent applications in drug design
2020 C. Bolchi, F. Bavo, R. Appiani, G. Roda, M. Pallavicini
Efficient One-Pot Reductive Aminations of Carbonyl Compounds with Aquivion-Fe as a Recyclable Catalyst and Sodium Borohydride
2020 V. Airoldi, O. Piccolo, G. Roda, R. Appiani, F. Bavo, R. Tassini, S. Paganelli, S. Arnoldi, M. Pallavicini, C. Bolchi
Behavioural and pharmacological profiles of zebrafish administrated pyrrolidinyl benzodioxanes and prolinol aryl ethers with high affinity for heteromeric nicotinic acetylcholine receptors
2020 D. Braida, L. Ponzoni, M. Moretti, P. Viani, M. Pallavicini, C. Bolchi, R. Appiani, F. Bavo, C. Gotti, M. Sala
SUBTYPE-SELECTIVE NEURONAL NICOTINIC ACETYLCHOLINE RECEPTOR AGONISTS AND ANTAGONISTS
2019 F. Bavo
Potent Antiglioblastoma Agents by Hybridizing the Onium-Alkyloxy-Stilbene Based Structures of an α7-nAChR, α9-nAChR Antagonist and of a Pro-Oxidant Mitocan
2018 F. Bavo, S. Pucci, F. Fasoli, C. Lammi, M. Moretti, V. Mucchietto, D. Lattuada, P. Viani, C. De Palma, R. Budriesi, I. Corradini, C. Dowell, J.M. Mcintosh, F. Clementi, C. Bolchi, C. Gotti, M. Pallavicini
Preparation of enantiopure methionine, arginine, tryptophan, and proline benzyl esters in green ethers by Fischer–Speier reaction
2018 C. Bolchi, F. Bavo, L. Regazzoni, M. Pallavicini
From pyrrolidinyl-benzodioxane to pyrrolidinyl-pyridodioxanes, or from unselective antagonism to selective partial agonism at alpha4beta2 nicotinic acetylcholine receptor
2017 C. Bolchi, F. Bavo, C. Gotti, L. Fumagalli, F. Fasoli, M. Binda, V. Mucchietto, M. Sciaccaluga, S. Plutino, S. Fucile, M. Pallavicini
Preparation and unequivocal identification of the regioisomers of nitrocatechol monobenzyl ether
2017 C. Bolchi, F. Bavo, M. Pallavicini
Molecular Hybridization of Potent and Selective γ-Hydroxybutyric Acid (GHB) Ligands: Design, Synthesis, Binding Studies, and Molecular Modeling of Novel 3-Hydroxycyclopent-1-enecarboxylic Acid (HOCPCA) and trans-γ-Hydroxycrotonic Acid (T-HCA) Analogs
2017 J. Krall, C.H. Jensen, F. Bavo, C.B. Falk-Petersen, A.S. Haugaard, S.B. Vogensen, Y. Tian, M. Nittegaard-Nielsen, S.B. Sigurdardã³ttir, J. Kehler, K.T. Kongstad, D.E. Gloriam, R.P. Clausen, K. Harpsã¸e, P. Wellendorph, B. Frølund
One-step preparation of enantiopure L- or D-amino acid benzyl esters avoiding the use of banned solvents
2017 C. Bolchi, F. Bavo, M. Pallavicini
Phase Diagrams to Evaluate the Opportunity for Enantiomeric Enrichment of Some Nonracemic Mixtures of Amino Acid Benzyl Esters by Crystallization as p-Toluenesulfonate Salts
2017 C. Bolchi, F. Bavo, M. Pallavicini
Structure Activity Relationship of novel antimicrobial agents, acting as inhibitors of the bacterial cell division protein Ftsz
2016 V. Straniero, C. Zanotto, L. Fumagalli, C. Bolchi, A. Radaelli, F. Bavo, M. Sanguinetti, C. De Giuli Morghen, M. Pallavicini
Novel 5-substituted 3-hydroxyphenyl and 3-nitrophenyl ethers of S-prolinol as α4β2-nicotinic acetylcholine receptor ligands
2016 C. Bolchi, F. Bavo, L. Fumagalli, C. Gotti, F. Fasoli, M. Moretti, M. Pallavicini
Crystallization-based resolution of 1,4-benzodioxane-2-carboxylic acid enantiomers via diastereomeric 1-phenylethylamides
2016 L. Fumagalli, C. Bolchi, F. Bavo, M. Pallavicini