Sfoglia per Autore
Regioselective Preparation of Functionalized Isoxazoline Derivatives, Key Intermediates in the Synthesis of Selective NMDA Receptor Antagonists
2011 L. Tamborini, A. Pinto, P. Conti, M. Gallanti, M.C. Iannuzzi, L. Lo Presti, C. De Micheli
Drug Discovery Targeting Amino Acid Racemases
2011 P. Conti, L. Tamborini, A. Pinto, A. Blondel, P. Minoprio, A. Mozzarelli, C. De Micheli
Synthesis and Biological Evaluation of CTP Synthetase Inhibitors as Potential Agents for the Treatment of African Trypanosomiasis
2012 L. Tamborini, A. Pinto, T.K. Smith, L.L. Major, M.C. Iannuzzi, S. Cosconati, L. Marinelli, E. Novellino, L. Lo Presti, P.E. Wong, M.P. Barrett, C. De Micheli, P. Conti
One-pot chemoenzymatic synthesis of aldoximes from primary alcohols in water
2012 P. Zambelli, A. Pinto, D. Romano, E. Crotti, P. Conti, L. Tamborini, R. Villa, F. Molinari
Ligand-exchange enantioresolution of dihydroisoxazole amino acid derivatives acting as glutamatergic modulators
2012 R. Sardella, F. Ianni, N. Giacchè, A. Lisanti, P. Conti, A. Pinto, L. Tamborini, B. Natalini
Evading Pgp activity in drug-resistant cancer cells : a structural and functional study of antitubulin furan metotica compounds
2012 T.L. Nguyen, M.R. Cera, A. Pinto, L. Lo Presti, E. Hamel, P. Conti, R. Gussio, P.D. Wulf
Two examples of high-efficient and green biotransformations
2012 D. Romano, L. Tamborini, A. Pinto, P. Zambelli, P. Conti, F. Molinari
Mechanism of inhibition of the glutamate transporter EAAC1 by the conformationally-constrained glutamate analog (+)-HIP-B
2012 R. Callender, A. Gameiro, A. Pinto, C. De Micheli, C. Grewer
An efficient method for the lipase-catalysed resolution and in-line purification of racemic flurbiprofen in a continuous-flow reactor
2012 L. Tamborini, D. Romano, A. Pinto, A. Bertolani, F. Molinari, P. Conti
3-Carboxy-pyrazolinalanine as a new scaffold for developing potent and selective NMDA receptor antagonists
2013 L. Tamborini, A. Pinto, F. Mastronardi, M.C. Iannuzzi, G. Cullia, B. Nielsen, C. De Micheli, P. Conti
Biotransformation with whole microbial systems in a continuous flow reactor : resolution of (RS)-flurbiprofen using Aspergillus oryzae by direct esterification with ethanol in organic solvent
2013 L. Tamborini, D. Romano, A. Pinto, M. Contente, M.C. Iannuzzi, P. Conti, F. Molinari
Inhibition of Rhodesain as a Novel Therapeutic Modality for Human African Trypanosomiasis
2013 R. Ettari, L. Tamborini, I.C. Angelo, N. Micale, A. Pinto, C. De Micheli, P. Conti
Pichia Glucozyma: a powerful biocatalyst for enantioselective reduction of ketones
2013 M.L. Contente, D. Romano, P. Conti, R. Gandolfi, A. Pinto, L. Tamborini, F. Molinari
Development of Rhodesain Inhibitors with a 3-Bromoisoxazoline Warhead
2013 R. Ettari, L. Tamborini, I.C. Angelo, S. Grasso, T. Schirmeister, L. Lo Presti, C. De Micheli, A. Pinto, P. Conti
Biotransformation of aromatic ketones and ketoesters with the non-conventional yeast Pichia glucozyma
2014 M.L. Contente, F. Molinari, P. Zambelli, V. De Vitis, R. Gandolfi, A. Pinto, D. Romano
Synthesis of (3-hydroxy-pyrazolin-5-yl)glycine based ligands interacting with ionotropic glutamate receptors
2014 A. Pinto, L. Tamborini, F. Mastronardi, R. Ettari, Y. Safoz, L. Bunch, B. Nielsen, A.A. Jensen, C. De Micheli, P. Conti
A new chemoenzymatic approach to the synthesis of latanoprost and bimatoprost
2014 D. Romano, M.L. Contente, F. Molinari, L. Tamborini, A. Pinto, P. Conti
Efficient synthesis of novel glutamate homologues and investigation of their affinity and selectivity profile at ionotropic glutamate receptors
2014 A. Pinto, L. Tamborini, F. Mastronardi, R. Ettari, D. Romano, B. Nielsen, C. De Micheli, P. Conti
Synthesis and biological evaluation of papain-family cathepsinl-like cysteine protease inhibitors containing a 1,4-benzodiazepine scaffold as antiprotozoal agents
2014 R. Ettari, A. Pinto, L. Tamborini, I.C. Angelo, S. Grasso, M. Zappalà, N. Capodicasa, L. Yzeiraj, E. Gruber, M.N. Aminake, G. Pradel, T. Schirmeister, C. De Micheli, P. Conti
Development of novel selective peptidomimetics containing a boronic acid moiety, targeting the 20s proteasome as anticancer agents
2014 K. Scarbaci, V. Troiano, R. Ettari, A. Pinto, N. Micale, C. Di Giovanni, C. Cerchia, T. Schirmeister, E. Novellino, A. Lavecchia, M. Zappalà, S. Grasso
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