Sfoglia per Autore
Progettazione e sintesi di nuovi agenti neuroprotettivi diretti verso il sistema glutammatergico
2008 P. Conti, A. Pinto, L. Tamborini, G. Grazioso, C. De Micheli
Neuroprotective effects of the novel glutamate transporter inhibitor (-)-3-hydroxy-4,5,6,6a-tetrahydro-3aH-pyrrolo[3,4-d]isoxazole-4-carboxylic acid, which preferentially inhibits reverse transport (glutamate release) compared with glutamate reuptake
2008 S. Colleoni, A.A. Jensen, E. Landucci, E. Fumagalli, P. Conti, A. Pinto, M. De Amici, D.E. Pellegrini Giampietro, C. De Micheli, T. Mennini, M. Gobbi
Synthesis and neuroprotective activity of new potent competitive NMDA receptor antagonists
2008 P. Conti, A. Pinto, L. Tamborini, E. Landucci, D.E. Pellegrini Giampietro, C. De Micheli
Synthesis and anti-HIV activity evaluation of new phenyl ethyl thiourea (PET) derivatives
2009 R. Ettari, A. Pinto, N. Micale
A regioselective route to 5-substituted isoxazoline-3-phosphonates
2009 P. Conti, A. Pinto, L. Tamborini, P. Dunkel, V. Gambaro, G.L. Visconti, C. De Micheli
A novel simplified synthesis of Acivicin
2009 A. Pinto, P. Conti, L. Tamborini, C. De Micheli
Synthesis of TBOA homologues and evaluation of their activity as Glutamate transporter inhibitors
2009 L. Tamborini, P. Conti, A. Pinto, M.C. Iannuzzi, C. De Micheli
Synthesis of new β- and γ-benzyloxy-S-glutamic acid derivatives and evaluation of their activity as inhibitors of excitatory amino acid transporters
2009 L. Tamborini, P. Conti, A. Pinto, S. Colleoni, M. Gobbi, C. De Micheli
Synthetic approach to and biological relevance of differently 3-subsituted delta2-isoxazolines and isoxazoles
2009 A. Pinto, L. Tamborini, P. Conti, C. De Micheli
A highly efficient flow reactor process for the synthesis of N-Boc-3,4-dehydro-L-proline methyl ester
2010 L. Tamborini, P. Conti, A. Pinto, C. De Micheli
Synthesis and biological evaluation of delta2—isoxazoline derivatives as DNA methyltransferase 1 inhibitors
2010 M. Viviano, S. Castellano, P. Conti, L. Tamborini, A. Pinto, S. Sicher, D. Kuck, C. De Micheli, J.L. Medina Franco, F. Lyko, G. Sbardella
CTP synthetase inhibitors as new potential agents for the treatment of African Trypanosomiasis : synthesis and in vitro/in vivo evaluation of trypanocidal activity of 3-Br-Acivicin
2010 P. Conti, A. Pinto, L. Tamborini, M.C. Iannuzzi, N. Patelli, C. De Micheli, M. Barrett, P.E. Wong, L.L. Major, T.K. Smith
SYNTHESIS AND BIOLOGICAL EVALUATION OF D2-ISOXAZOLINE DERIVATIVES AS DNA METHYLTRANSFERASE 1 INHIBITORS
2010 M. Viviano, S. Castellano, P. Conti, L. Tamborini, A. Pinto, S. Sicher, D. Kuck, C. DE MICHELI, J.L. MEDINA FRANCO, F. Lyko, G. Sbardella
Design and synthesis of novel isoxazole-based HDAC inhibitors
2010 P. Conti, L. Tamborini, A. Pinto, L. Sola, R. Ettari, C. Mercurio, C. De Micheli
Novel 3-carboxy- and 3-phosphono-pyrazoline amino acids acting as potent and selective NMDA receptor antagonists: design, synthesis and pharmacological characterization
2010 P. Conti, A. Pinto, L. Tamborini, U. Madsen, B. Nielsen, H. Bräuner Osborne, K.B. Hansen, E. Landucci, D.E. Pellegrini Giampietro, G. De Sarro, E. Donato Di Paola, C. De Micheli
Synthesis of 3-Aryl/benzyl-4,5,6,6a-tetrahydro-3aHpyrrolo[3,4-d]isoxazole Derivatives: A Comparison between Conventional, Microwave-Assisted and Flow-Based Methodologies
2010 S. Castellano, L. Tamborini, M. Viviano, A. Pinto, G. Sbardella, P. Conti
From potent AMPA/KA agonists to either selective NMDA antagonists or to inhibitors of the glutamate transporters
2011 C. De Micheli, P. Conti, A. Pinto, L. Tamborini
Synthesis of new isoxazoline-based acidic amino acids and investigation of their affinity and selectivity profile at ionotropic glutamate receptors
2011 A. Pinto, P. Conti, G. Grazioso, L. Tamborini, U. Madsen, B. Nielsen, C. De Micheli
Synthesis and Biochemical Evaluation of Δ2-Isoxazoline Derivatives as DNA Methyltransferase 1 Inhibitors
2011 S. Castellano, D. Kuck, M. Viviano, J. Yoo, F. López-Vallejo, P. Conti, L. Tamborini, A. Pinto, J.L. Medina-Franco, G. Sbardella
Synthesis and in vitro/in vivo Evaluation of the Antitrypanosomal Activity of 3-Bromoacivicin, a Potent CTP Synthetase Inhibitor
2011 P. Conti, A. Pinto, P.E. Wong, L.L. Major, L. Tamborini, M.C. Iannuzzi, C. De Micheli, M.P. Barrett, T.K. Smith
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