Sfoglia per Autore
Optimization of peptidomimetic boronates bearing a P3 bicyclic scaffold as proteasome inhibitors
2014 V. Troiano, K. Scarbaci, R. Ettari, N. Micale, C. Cerchia, A. Pinto, T. Schirmeister, E. Novellino, S. Grasso, A. Lavecchia, M. Zappalà
Discovery of covalent inhibitors of glyceraldehyde-3-phosphate dehydrogenase, a target for the treatment of malaria
2014 S. Bruno, A. Pinto, G. Paredi, L. Tamborini, C. De Micheli, V. La Pietra, L. Marinelli, E. Novellino, P. Conti, A. Mozzarelli
Rationalizing the Lacking of Inversion Symmetry in a Noncentrosymmetric Polar Racemate : an Experimental and Theoretical Study
2014 L. Lo Presti, M. Sist, L. Loconte, A. Pinto, L. Tamborini, C. Gatti
Use of a O-benzyl-(S)-serine containing eluent for the efficient ligand-exchange chromatography-based enantioseparation of constrained glutamate receptor ligands
2015 F. Ianni, R. Sardella, A. Lisanti, N. Giacchè, P. Conti, A. Pinto, L. Tamborini, B. Natalini
A new chemoenzymatic approach to the synthesis of Latanoprost and Bimatoprost
2015 M. Contente, P. Zambelli, S. Galafassi, L. Tamborini, A. Pinto, P. Conti, F. Molinari, D. Romano
Synthesis and Pharmacological Evaluation of (42) Nicotinic Ligands with a 3-Fluoropyrrolidine Nucleus
2015 L. Tamborini, A. Pinto, R. Ettari, C. Gotti, F. Fasoli, P. Conti, C. Demicheli
Synthesis of unusual isoxazoline containing β and γ-dipeptides as potential glutamate receptor ligands
2015 L. Tamborini, F. Mastronardi, F. Dall'Oglio, C. De Micheli, B. Nielsen, L. Lo Presti, P. Conti, A. Pinto
Stereoselective reduction of aromatic ketones by a new ketoreductase from Pichia glucozyma
2015 M.L. Contente, D. Romano, I. Eberini, A. Pinto, F.E. Molinari
Characterization of 2,4-Diamino-6-oxo-1,6-dihydropyrimidin-5-yl Ureido Based Inhibitors of Trypanosoma brucei FolD and Testing for Antiparasitic Activity
2015 T.C. Eadsforth, A. Pinto, R. Luciani, L. Tamborini, G. Cullia, C. De Micheli, L. Marinelli, S. Cosconati, E. Novellino, L. Lo Presti, A. Cordeiro da Silva, P. Conti, W.N. Hunter, M.P. Costi
Development of novel dipeptide-like rhodesain inhibitors containing the 3-bromoisoxazoline warhead in a constrained conformation
2015 R. Ettari, A. Pinto, S. Previti, L. Tamborini, I..C. Angelo, V. La Pietra, L. Marinelli, E. Novellino, T. Schirmeister, M. Zappalà, S. Grasso, C. De Micheli, P. Conti
Enzymatic reduction of acetophenone derivatives with a benzil reductase from Pichia glucozyma (KRED1-Pglu): electronic and steric effects on activity and enantioselectivity
2016 M.L. Contente, I. Serra, L. Palazzolo, C. Parravicini, E. Gianazza, I. Eberini, A. Pinto, B. Guidi, F. Molinari, D. Romano
Stereoselective Enzymatic Reduction of Ethyl Secodione : Preparation of a Key Intermediate for the Total Synthesis of Steroids
2016 M.L. Contente, F. Molinari, I. Serra, A. Pinto, D. Romano
γ-Glutamyl-dipeptides : Easy tools to rapidly probe the stereoelectronic properties of the ionotropic glutamate receptor binding pocket
2016 L. Tamborini, V. Nicosia, P. Conti, F. Dall'Oglio, C. De Micheli, B. Nielsen, A.A. Jensen, D.S. Pickering, A. Pinto
Selectivity of 3-bromo-isoxazoline inhibitors between human and Plasmodium falciparum glyceraldehyde-3-phosphate dehydrogenases
2016 S. Bruno, M. Margiotta, A. Pinto, G. Cullia, P. Conti, C. De Micheli, A. Mozzarelli
An efficient continuous flow process for the synthesis of a non-conventional mixture of fructooligosaccharides
2016 P. Zambelli, L. Tamborini, S. Cazzamalli, A. Pinto, S. Arioli, S. Balzaretti, F.J. Plou, L. Fernandez Arrojo, F. Molinari, P. Conti, D. Romano
Inspired by Nature : The 3-Halo-4,5-dihydroisoxazole Moiety as a Novel Molecular Warhead for the Design of Covalent Inhibitors
2016 A. Pinto, L. Tamborini, G. Cullia, P. Conti, C. De Micheli
Bicyclic γ-amino acids as inhibitors of γ-aminobutyrate aminotransferase
2016 A. Pinto, L. Tamborini, E. Pennacchietti, A. Coluccia, R. Silvestri, G. Cullia, C. De Micheli, P. Conti, D. De Biase
Synthesis and biological evaluation of new ligands designed to selectively interact with kainate receptors
2016 G. Cullia, F. Mastronardi, A. Pinto, L. Tamborini, L. Marconi, C. De Micheli, P. Conti
Preparation of enantiomerically enriched aromatic β-hydroxynitriles and halohydrins by ketone reduction with recombinant ketoreductase KRED1-Pglu
2016 M.L. Contente, I. Serra, F. Molinari, R. Gandolfi, A. Pinto, D. Romano
The chemoenzymatic continuous-flow synthesis of captopril
2016 F. Dall'Oglio, A. Pinto, V. De Vitis, F. Molinari, D. Romano, P. Conti, L. Tamborini
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