DE MICHELI, CARLO
DE MICHELI, CARLO
Dipartimento di Scienze Farmaceutiche
Folates in Trypanosoma brucei: achievements and opportunities
2018 G. Cullia, L. Tamborini, P. Conti, C. De Micheli, A. Pinto
Effects of 3-bromo-4,5-dihydroisoxazole derivatives on Nrf2 activation and heme oxygenase-1 expression
2018 A. Pinto, Z. El Ali, S. Moniot, L. Tamborini, C. Steegborn, R. Foresti, C. De Micheli
Flow-based biocatalysis : application to peracetylated arabinofuranosyl-1,5-arabinofuranose synthesis
2018 T. Bavaro, A. Pinto, F. Dall'Oglio, M.J. Hernaiz, C.F. Morelli, P. Zambelli, C. De Micheli, P. Conti, L. Tamborini, M. Terreni
Chemoenzymatic synthesis in flow reactors: a rapid and convenient preparation of Captopril
2017 V. De Vitis, F. Dall’Oglio, A. Pinto, C. De Micheli, F.E. Molinari, P. Conti, D. Romano, L. Tamborini
Structural basis of subunit-selectivity for competitive NMDA receptor antagonists with preference for GluN2A over GluN2B subunits
2017 G.E. Lind, T.-.C. Mou, L. Tamborini, M.G. Pomper, C. De Micheli, P. Conti, A. Pinto, K.B. Hansen
Synthesis of L-tricholomic acid analogues and pharmacological characterization at ionotropic glutamate receptors
2017 L. Tamborini, F. Mastronardi, L. Lo Presti, B. Nielsen, C. De Micheli, P. Conti, A. Pinto
Design, synthesis and biological characterization of PfGAPDH inhibitors
2016 G. Cullia, A. Pinto, S. Bruno, S. Parapini, L. Tamborini, A. Mozzarelli, D. Taramelli, C. De Micheli, P. Conti
Synthesis and pharmacological evaluation of conformationally constrained glutamic acid higher homologues
2016 L. Tamborini, G. Cullia, B. Nielsen, C. De Micheli, P. Conti, A. Pinto
Development of Radiolabeled Ligands Targeting the Glutamate Binding Site of the N-Methyl-d-aspartate Receptor as Potential Imaging Agents for Brain
2016 L. Tamborini, Y. Chen, C.A. Foss, A. Pinto, A.G. Horti, S.F. Traynelis, C. De Micheli, R.C. Mease, K.B. Hansen, P. Conti, M.G. Pomper
Synthesis and biological evaluation of new ligands designed to selectively interact with kainate receptors
2016 G. Cullia, F. Mastronardi, A. Pinto, L. Tamborini, L. Marconi, C. De Micheli, P. Conti
Selectivity of 3-bromo-isoxazoline inhibitors between human and Plasmodium falciparum glyceraldehyde-3-phosphate dehydrogenases
2016 S. Bruno, M. Margiotta, A. Pinto, G. Cullia, P. Conti, C. De Micheli, A. Mozzarelli
Inspired by Nature : The 3-Halo-4,5-dihydroisoxazole Moiety as a Novel Molecular Warhead for the Design of Covalent Inhibitors
2016 A. Pinto, L. Tamborini, G. Cullia, P. Conti, C. De Micheli
γ-Glutamyl-dipeptides : Easy tools to rapidly probe the stereoelectronic properties of the ionotropic glutamate receptor binding pocket
2016 L. Tamborini, V. Nicosia, P. Conti, F. Dall'Oglio, C. De Micheli, B. Nielsen, A.A. Jensen, D.S. Pickering, A. Pinto
Bicyclic γ-amino acids as inhibitors of γ-aminobutyrate aminotransferase
2016 A. Pinto, L. Tamborini, E. Pennacchietti, A. Coluccia, R. Silvestri, G. Cullia, C. De Micheli, P. Conti, D. De Biase
Development of novel dipeptide-like rhodesain inhibitors containing the 3-bromoisoxazoline warhead in a constrained conformation
2015 R. Ettari, A. Pinto, S. Previti, L. Tamborini, I..C. Angelo, V. La Pietra, L. Marinelli, E. Novellino, T. Schirmeister, M. Zappalà, S. Grasso, C. De Micheli, P. Conti
Synthesis of unusual isoxazoline containing β and γ-dipeptides as potential glutamate receptor ligands
2015 L. Tamborini, F. Mastronardi, F. Dall'Oglio, C. De Micheli, B. Nielsen, L. Lo Presti, P. Conti, A. Pinto
Synthesis and Pharmacological Evaluation of (42) Nicotinic Ligands with a 3-Fluoropyrrolidine Nucleus
2015 L. Tamborini, A. Pinto, R. Ettari, C. Gotti, F. Fasoli, P. Conti, C. Demicheli
Characterization of 2,4-Diamino-6-oxo-1,6-dihydropyrimidin-5-yl Ureido Based Inhibitors of Trypanosoma brucei FolD and Testing for Antiparasitic Activity
2015 T.C. Eadsforth, A. Pinto, R. Luciani, L. Tamborini, G. Cullia, C. De Micheli, L. Marinelli, S. Cosconati, E. Novellino, L. Lo Presti, A. Cordeiro da Silva, P. Conti, W.N. Hunter, M.P. Costi
Synthesis and biological evaluation of papain-family cathepsinl-like cysteine protease inhibitors containing a 1,4-benzodiazepine scaffold as antiprotozoal agents
2014 R. Ettari, A. Pinto, L. Tamborini, I.C. Angelo, S. Grasso, M. Zappalà, N. Capodicasa, L. Yzeiraj, E. Gruber, M.N. Aminake, G. Pradel, T. Schirmeister, C. De Micheli, P. Conti
Synthesis of (3-hydroxy-pyrazolin-5-yl)glycine based ligands interacting with ionotropic glutamate receptors
2014 A. Pinto, L. Tamborini, F. Mastronardi, R. Ettari, Y. Safoz, L. Bunch, B. Nielsen, A.A. Jensen, C. De Micheli, P. Conti