PARAPINI, SILVIA
PARAPINI, SILVIA
Dipartimento di Scienze Biomediche per la Salute
Novel antimalarial 3-substituted quinolones isosteres with improved pharmacokinetic properties
2025 S. Ge, R. Jian, Q. Xuan, Y. Zhu, X. Ren, W. Li, X. Chen, R.K. Huang, C.S. Lee, S.C. Leung, N. Basilico, S. Parapini, D. Taramelli, N. Pinthong, S.V. Antonyuk, P.M. O'Neill, Z. Sheng, W.D. Hong
From pan-active to parasite-selective antiparasitic agents: A scaffold hopping approach
2025 C. Borsari, N. Santarem, D. Coertzen, A. Mazzolari, A.I. Corfu, C. Coelho, F. Barbosa, L. Tamborini, L.-. Birkholtz, L. Raffellini, O. Keminer, N. Basilico, S. Parapini, S. Gul, A. Cordeiro-da-Silva, P. Conti
Two-Step Flow Amidation of Natural Phenolic Acids as Antiradical and Antimicrobial Agents
2025 D. Pecora, A.M. Magni, S. Vicinanza, F. Annunziata, S. Princiotto, S. Donzella, G. Meroni, P.A. Martino, N. Basilico, S. Parapini, P. Conti, C. Borsari, L. Tamborini
Antiprotozoal Activity of Highly Substituted Pyrazole and Pyrimidine Derivatives
2025 M. Lusardi, N. Basilico, E. Iervasi, C. Brullo, S. Parapini, M. Ponassi, C. Rosano, A. Spallarossa
Discovery of 1,3,4-Oxadiazole Derivatives as Broad-Spectrum Antiparasitic Agents
2024 A.I. Corfu, N. Santarem, S. Luelmo, G. Mazza, A. Greco, A. Altomare, G. Ferrario, G. Nasta, O. Keminer, G. Aldini, L. Tamborini, N. Basilico, S. Parapini, S. Gul, A. Cordeiro-da-Silva, P. Conti, C. Borsari
Design, synthesis and modelling of photoreactive chemical probes for investigating target engagement of plasmepsin IX and X in Plasmodium falciparum
2024 M. Lisauskaitė, G.L. Nixon, C.M. Woodley, N.G. Berry, A. Coninckx, L. Charlie Qie, S.C. Leung, D. Taramelli, N. Basilico, S. Parapini, S.A. Ward, O. Vadas, D. Soldati-Favre, W. David Hong, P.M. O'Neill
Screening of Mpro Protease (SARS-CoV-2) Covalent Inhibitors from an Anthocyanin-Rich Blueberry Extract Using an HRMS-Based Analytical Platform
2024 A. Altomare, G. Baron, G. Cambiaghi, G. Ferrario, B. Zoanni, L. Della Vedova, G.M. Fumagalli, S. D'Alessandro, S. Parapini, S. Vittorio, G. Vistoli, P. Riso, M. Carini, S. Delbue, G. Aldini
In Vitro Screening of an In-House Library of Structurally Distinct Chemotypes Towards the Identification of Novel SARS-CoV-2 Inhibitors
2024 M. Tonelli, A. Sparatore, I. Bassanini, V. Francesconi, F. Sparatore, K.K. Maina, S. Delbue, S. D'Alessandro, S. Parapini, N. Basilico
Novel chemo-enzymatic synthesis, structural elucidation and first antiprotozoal activity profiling of the atropoisomeric dimers of trans-8-Hydroxycalamenene
2024 I. Bassanini, C. Tognoli, M. Meli, S. Parapini, N. Basilico, G. Fronza, S. Serra, S. Riva
Multiplex array analysis of circulating cytokines and chemokines in COVID-19 patients during the first wave of the SARS-CoV-2 pandemic in Milan, Italy
2024 E. Calvo-Alvarez, S. D'Alessandro, N. Zanotta, N. Basilico, S. Parapini, L. Signorini, F. Perego, K.K. Maina, P. Ferrante, A. Modenese, P. Pizzocri, A. Ronsivalle, S. Delbue, M. Comar
A ChemoEnzymatic Approach for the Preparation of “Linear-Shaped” Diaryl Pyrazines as Potential Antiprotozoal Agents
2024 I. Bassanini, T. Braga, C. Tognoli, M. Vanoni, G. Mazza, N. Basilico, S. Parapini, S. Riva
Role of Stereochemistry on the Biological Activity of Nature-Inspired 3-Br-Acivicin Isomers and Derivatives
2023 A. Galbiati, A. Zana, C. Borsari, M. Persico, S. Bova, O. Tkachuk, A.I. Corfu, L. Tamborini, N. Basilico, C. Fattorusso, S. Bruno, S. Parapini, P. Conti
Heat-Treated Lysozyme Hydrochloride: A Study on Its Structural Modifications and Anti-SARS-CoV-2 Activity
2023 S. Delbue, E. Pariani, S. Parapini, C. Galli, N. Basilico, S. D’Alessandro, S. Pellegrino, E. Pini, S. Ciceri, P. Ferraboschi, P. Grisenti
Antimalarial Activity of Tri- and Tetra-Substituted Anilino Pyrazoles
2023 M. Lusardi, N. Basilico, C. Rotolo, S. Parapini, A. Spallarossa
Efficient One-Pot Synthesis of Novel Caffeic Acid Derivatives as Potential Antimalarials
2023 K. Sidoryk, S. Parapini, N. Basilico, M. Zaremba-Czogalla, M. Kubiszewski, M. Cybulski, J. Gubernator, A. Zagórska, A. Jaromin
Favorable Preclinical Pharmacological Profile of a Novel Antimalarial Pyrrolizidinylmethyl Derivative of 4-amino-7-chloroquinoline with Potent In Vitro and In Vivo Activities
2023 N. Basilico, S. Parapini, S. D’Alessandro, P. Misiano, S. Romeo, G. Dondio, V. Yardley, L. Vivas, S. Nasser, L. Rénia, B.M. Russell, R. Suwanarusk, F. Nosten, A. Sparatore, D. Taramelli
In Vitro Antiparasitic Activities of Monovalent Ionophore Compounds for Human and Canine Leishmaniases
2022 E. Calvo Alvarez, S. D'Alessandro, D. Proverbio, E. Spada, R. Perego, D. Taramelli, N. Basilico, S. Parapini
Eco design for Ag-based solutions against SARS-CoV-2 and E. coli
2022 A.L. Costa, M. Blosi, A. Brigliadori, I. Zanoni, S. Ortelli, F.C. Simeone, S. Delbue, S. D'Alessandro, S. Parapini, C. Vineis, A. Varesano, M.S. Toprak, B. Hamawandi, D. Gardini
Total Synthesis of the Natural Chalcone Lophirone E, Synthetic Studies toward Benzofuran and Indole-Based Analogues, and Investigation of Anti-Leishmanial Activity
2022 L. Pozzetti, R. Ibba, S. Rossi, O. Taglialatela-Scafati, D. Taramelli, N. Basilico, S. D'Alessandro, S. Parapini, S. Butini, G. Campiani, S. Gemma
A rapid spectrophotometric method to identify inhibitors of human erythropoiesis
2022 D.P. Ilboudo, S. D'Alessandro, S. Parapini, E.C. Alvarez, P. Misiano, D. Taramelli, N. Basilico