Sfoglia per Autore
Targeting integrins alphaVbeta3 and alphaIIbeta3 with RGD peptidomimetics : study of the ligand conformation and of the ligand-receptor interactions
2011 M. Civera, L. Belvisi, C. Gennari, U. Piarulli, D. Potenza, F. Vasile
RGD-based peptides targheting αIIbβ3 and αvβ3 integrin receptors: an NMR point of view
2011 D. Potenza, F. Vasile, L. Belvisi, M. Civera, L. Colombo, M. Serra
Ligand-target interaction: a NMR point of view
2012 D. Potenza, F. Vasile
Dimeric Smac mimetics/IAP inhibitors as in vivo-active pro-apoptotic agents. Part II : Structural and biological characterization
2012 D. Lecis, E. Mastrangelo, L. Belvisi, M. Bolognesi, M. Civera, F. Cossu, M. De Cesare, D. Delia, C. Drago, G. Manenti, L. Manzoni, M. Milani, E. Moroni, P. Perego, D. Potenza, V. Rizzo, C. Scavullo, C. Scolastico, F. Servida, F. Vasile, P. Seneci
Design, Synthesis and Biological Evaluation of Novel cRGD-Paclitaxel Conjugates for Integrin-Assisted Drug Delivery
2012 M. Pilkington-Miksa, D. Arosio, L. Battistini, L. Belvisi, M. De Matteo, F. Vasile, P. Burreddu, P. Carta, G. Rassu, P. Perego, N. Carenini, F. Zunino, M. De Cesare, V. Castiglioni, E. Scanziani, C. Scolastico, G. Casiraghi, F. Zanardi, L. Manzoni
A NMR and computational study of Smac mimics targeting both the BIR2 and BIR3 domains in XIAP protein
2012 D. Potenza, L. Belvisi, F. Vasile, E. Moroni, F. Cossu, P. Seneci
Homo- and heterodimeric Smac mimetics/IAP inhibitors as in vivo-active pro-apoptotic agents. Part I : synthesis
2012 L. Manzoni, L. Belvisi, A. Bianchi, A. Conti, C. Drago, M. de Matteo, L. Ferrante, E. Mastrangelo, P. Perego, D. Potenza, C. Scolastico, F. Servida, G. Timpano, F. Vasile, V. Rizzo, P. Seneci
Solution structure by nuclear magnetic resonance of the two lantibiotics 97518 and NAI-107
2012 F. Vasile, D. Potenza, B. Marsiglia, S. Maffioli, S. Donadio
Both El Tor and classical cholera toxin bind blood group determinants
2012 J. E. Heggelund, E. Haugen, B. Lygren, A. Mackenzie, Å. Holmner, F. Vasile, J.J. Reina Martin, A. Bernardi, U. Krengel
Cyclic RGD Peptidomimetics Containing Bifunctional Diketopiperazine Scaffolds as New Potent Integrin Ligands
2012 M. Marchini, M. Mingozzi, R. Colombo, I. Guzzetti, L. Belvisi, F. Vasile, D. Potenza, U. Piarulli, D. Arosio, C.M.A. Gennari
Determination of the binding epitope of RGD-peptidomimetics to αvβ3 and αIIbβ3 integrin-rich intact cells by NMR and computational studies
2013 I. Guzzetti, M. Civera, F. Vasile, E.M.V. Araldi, L. Belvisi, C.M.A. Gennari, D. Potenza, R. Fanelli, U. Piarulli
New homo- and heretodimeric SMAC mimetic compound as apoptosis inducers
2013 P. Seneci, L. Belvisi, F. Cossu, D. Delia, C. Drago, D. Lecis, S. Maiorana, L.P. Manzoni, E. Mastrangelo, M. Milani De Mayo De Mari, P.M.C. Perego, F. Vasile
STD-NMR experiments on tumor cells to investigate RGD ligand - membrane protein interactions
2013 I. Guzzetti, D. Potenza, F. Vasile, L. Belvisi, M. Civera, I. Silvestri, U. Piarulli, C. Gennari
A Comprehensive NMR Analysis of the Interaction between DKP-RGD Ligands and Membrane Proteins on Intact Cells
2013 I. Guzzetti, D. Potenza, F. Vasile, L. Belvisi, M. Civera, I. Silvestri, U. Piarulli, C. Gennari
Comprehensive analysis of blood group antigen binding to classical and El Tor cholera toxin B-pentamers by NMR
2014 F. Vasile, J.J. Reina, D. Potenza, J.E. Heggelund, A. Mackenzie, U. Krengel, A. Bernardi
Antitumor activity of a novel homodimeric SMAC mimetic in ovarian carcinoma
2014 L. Gatti, M. De Cesare, E. Ciusani, E. Corna, N. Arrighetti, D. Cominetti, L. Belvisi, D. Potenza, E. Moroni, F. Vasile, D. Lecis, D. Delia, V. Castiglioni, E. Scanziani, P. Seneci, N. Zaffaroni, P. Perego
Diffusion-ordered spectroscopy and saturation transfer difference NMR spectroscopy studies of selective interactions between ELAV protein fragments and an mRNA target
2014 F. Vasile, D. Rossi, S. Collina, D. Potenza
Cyclic RGD peptidomimetics: insights into the binding to integrin-rich cancer cells by NMR and computational studies
2015 L. Belvisi, D. Arosio, M. Civera, C. Gennari, I. Guzzetti, U. Piarulli, F. Vasile, D. Potenza
Synthesis of Functionalized 2-(4-Hydroxyphenyl)-3-methylbenzofuran Allosteric Modulators of Hsp90 Activity
2016 S. Sattin, M. Panza, F. Vasile, F. Berni, G. Goti, J. Tao, E. Moroni, D. Agard, G. Colombo, A. Bernardi
Different behavior of cyclic RGD peptidomimetics versus a5b1 and aVb3 integrin-rich cancer cells: NMR and computational analysis
2016 F. Vasile, M. Civera, D. Arosio, L. Belvisi, C. Gennari, U. Piarulli, D. Potenza
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