GENNARI, CESARE MARIO ARTURO
GENNARI, CESARE MARIO ARTURO
Dipartimento di Chimica
Amine-Carbamate Self-Immolative Spacers Counterintuitively Release 3° Alcohol at Much Faster Rates than 1° Alcohol Payloads
2024 M. Mason, L. BISBAL LOPEZ, F. Bashiri, A. Herrero, A. Baron, R. Bucci, L. Pignataro, C. Gennari, A. DAL CORSO
Ex vivo mass spectrometry-based biodistribution analysis of an antibody-Resiquimod conjugate bearing a protease-cleavable and acid-labile linker
2023 L. BISBAL LOPEZ, D. Ravazza, M. Bocci, A. Zana, L. Principi, S. Dakhel Plaza, A. Galbiati, E. Gilardoni, J. Scheuermann, D. Neri, L. Pignataro, C. Gennari, S. Cazzamalli, A. DAL CORSO
Visible Light-Promoted β-Functionalization of Carbonyl Compounds in the Presence of Organic Dyes
2023 L. Dolcini, T. Gandini, R. Castiglioni, A. Bossi, M. Penconi, A. DAL CORSO, C. Gennari, L. Pignataro
RGD cyclopeptide equipped with a lysine-engaging salicylaldehyde shows enhanced integrin affinity and cell detachment potency
2023 G. Sacco, D. Arosio, M. Paolillo, A. Gloger, J. Scheuermann, L.L. Pignataro, L. Belvisi, A. DAL CORSO, C.M.A. Gennari
Regiodivergent Reductive Opening of Epoxides by Catalytic Hydrogenation Promoted by a (Cyclopentadienone)iron Complex
2022 L. Tadiello, T. Gandini, B.M. Stadler, S. Tin, H. Jiao, J.G. de Vries, L.L. Pignataro, C.M.A. Gennari
Development and Biochemical Characterization of Self-Immolative Linker Containing GnRH-III-Drug Conjugates
2022 S. Schuster, É. Juhász, G. Halmos, I. Neundorf, C. Gennari, G. Mező
Advanced Pyrrolidine-Carbamate Self-Immolative Spacer with Tertiary Amine Handle Induces Superfast Cyclative Drug Release
2022 A. Dal Corso, M. Frigoli, M. Prevosti, M. Mason, R. Bucci, L. Belvisi, L. Pignataro, C. Gennari
Metallaphotoredox C-O and C-N Cross-coupling using Donor-Acceptor Cyanoarene Photocatalysts
2022 T. Gandini, L. Dolcini, L. Di Leo, M. Fornara, A. Bossi, M. Penconi, A. Dal Corso, C. Gennari, L. Pignataro
Functionalized 2-Hydroxybenzaldehyde-PEG Modules as Portable Tags for the Engagement of Protein Lysine ϵ-Amino Groups
2021 G. Sacco, S. Stammwitz, L. Belvisi, L. Pignataro, A. Dal Corso, C. Gennari
A Trifunctional Self-Immolative Spacer Enables Drug Release with Two Non-Sequential Enzymatic Cleavages
2021 A. DAL CORSO, S. Arosio, N. Arrighetti, P. Perego, L. Belvisi, L.L. Pignataro, C.M.A. Gennari
Celebrating Franco Cozzi's 70 th Birthday
2021 M. Benaglia, C. Gennari
Fast Cyclization of a Proline-Derived Self-Immolative Spacer Improves the Efficacy of Carbamate Prodrugs
2020 A. DAL CORSO, V. Borlandelli, C. Corno, P. Perego, L. Belvisi, L.L. Pignataro, C.M.A. Gennari
Multimeric Presentation of RGD Peptidomimetics Enhances Integrin Binding and Tumor Cell Uptake
2020 A. Pina, M. Kadri, D. Arosio, A. Dal Corso, J. Coll, C. Gennari, D. Boturyn
Recent Catalytic Applications of (Cyclopentadienone)iron Complexes
2020 L. Pignataro, C. Gennari
Synthesis and Biological Evaluation of RGD and isoDGR-Monomethyl Auristatin Conjugates Targeting Integrin αVβ3
2019 A. Raposo Moreira Dias, L. Bodero, A. Martins, D. Arosio, S. Gazzola, L. Belvisi, L. Pignataro, C. Steinkühler, A. Dal Corso, C. Gennari, U. Piarulli
Improving C=N Bond Reductions with (Cyclopentadienone)iron Complexes: Scope and Limitations
2019 M. Cettolin, X. Bai, D. Lübken, M. Gatti, S. Vailati Facchini, U. Piarulli, L. Pignataro, C. Gennari
Chiral (cyclopentadienone)iron complexes with a stereogenic plane as pre-catalysts for the asymmetric hydrogenation of polar double bonds
2019 X. Bai, M. Cettolin, G. Mazzoccanti, M. Pierini, U. Piarulli, V. Colombo, A. Dal Corso, L. Pignataro, C. Gennari
Hydrogen-Borrowing Amination of Secondary Alcohols Promoted by a (Cyclopentadienone)iron Complex
2019 X. Bai, F. Aiolfi, M. Cettolin, U. Piarulli, A. DAL CORSO, L.L. Pignataro, C.M.A. Gennari
β-Glucuronidase triggers extracellular MMAE release from an integrin-targeted conjugate
2019 P. López Rivas, C. Müller, C. Breunig, T. Hechler, A. Pahl, D. Arosio, L. Belvisi, L. Pignataro, A. Dal Corso, C. Gennari
Conjugates of Cryptophycin and RGD or isoDGR Peptidomimetics for Targeted Drug Delivery
2019 A. Borbély, E. Figueras, A. Martins, L. Bodero, A. Raposo moreira dias, P. López rivas, A. Pina, D. Arosio, P. Gallinari, M. Frese, C. Steinkühler, C. Gennari, U. Piarulli, N. Sewald