ETTARI, ROBERTA
ETTARI, ROBERTA
Dipartimento di Scienze Farmaceutiche
Development of novel dipeptide-like rhodesain inhibitors containing the 3-bromoisoxazoline warhead in a constrained conformation
2015 R. Ettari, A. Pinto, S. Previti, L. Tamborini, I..C. Angelo, V. La Pietra, L. Marinelli, E. Novellino, T. Schirmeister, M. Zappalà, S. Grasso, C. De Micheli, P. Conti
Synthesis and biological evaluation of papain-family cathepsinl-like cysteine protease inhibitors containing a 1,4-benzodiazepine scaffold as antiprotozoal agents
2014 R. Ettari, A. Pinto, L. Tamborini, I.C. Angelo, S. Grasso, M. Zappalà, N. Capodicasa, L. Yzeiraj, E. Gruber, M.N. Aminake, G. Pradel, T. Schirmeister, C. De Micheli, P. Conti
Development of novel selective peptidomimetics containing a boronic acid moiety, targeting the 20s proteasome as anticancer agents
2014 K. Scarbaci, V. Troiano, R. Ettari, A. Pinto, N. Micale, C. Di Giovanni, C. Cerchia, T. Schirmeister, E. Novellino, A. Lavecchia, M. Zappalà, S. Grasso
Synthesis of (3-hydroxy-pyrazolin-5-yl)glycine based ligands interacting with ionotropic glutamate receptors
2014 A. Pinto, L. Tamborini, F. Mastronardi, R. Ettari, Y. Safoz, L. Bunch, B. Nielsen, A.A. Jensen, C. De Micheli, P. Conti
Identification of a new series of amides as non-covalent proteasome inhibitors
2014 K. Scarbaci, V. Troiano, N. Micale, R. Ettari, L. Tamborini, C. Di Giovanni, C. Cerchia, S. Grasso, E. Novellino, T. Schirmeister, A. Lavecchia, M. Zappalà
Optimization of peptidomimetic boronates bearing a P3 bicyclic scaffold as proteasome inhibitors
2014 V. Troiano, K. Scarbaci, R. Ettari, N. Micale, C. Cerchia, A. Pinto, T. Schirmeister, E. Novellino, S. Grasso, A. Lavecchia, M. Zappalà
Efficient synthesis of novel glutamate homologues and investigation of their affinity and selectivity profile at ionotropic glutamate receptors
2014 A. Pinto, L. Tamborini, F. Mastronardi, R. Ettari, D. Romano, B. Nielsen, C. De Micheli, P. Conti
NMR Characterization and conformational analysis of a potent papain-family cathepsin L-like cysteine protease inhibitor with different behaviour in polar and apolar media
2014 A. Rotondo, R. Ettari, M. Zappalà, C. De Micheli, E. Rotondo
Synthesis of new 2-amino-6-(trifluoromethoxy)benzoxazole derivatives, analogues of riluzole
2013 M.L. Calabrò, R. Caputo, R. Ettari, G. Puia, F. Ravazzini, M. Zappalà, N. Micale
Development of Rhodesain Inhibitors with a 3-Bromoisoxazoline Warhead
2013 R. Ettari, L. Tamborini, I.C. Angelo, S. Grasso, T. Schirmeister, L. Lo Presti, C. De Micheli, A. Pinto, P. Conti
Efficient synthesis of kainic acid analogues
2013 L. Tamborini, F. Mastronardi, G. Cullia, R. Ettari, C. De Micheli
Development of Peptidomimetic Boronates as Proteasome Inhibitors
2013 N. Micale, R. Ettari, A. Lavecchia, C. Di Giovanni, K. Scarbaci, V. Troiano, S. Grasso, E. Novellino, T. Schirmeister, M. Zappalà
Inhibition of Rhodesain as a Novel Therapeutic Modality for Human African Trypanosomiasis
2013 R. Ettari, L. Tamborini, I.C. Angelo, N. Micale, A. Pinto, C. De Micheli, P. Conti
Synthesis and Molecular Modeling Studies of Derivatives of a Highly Potent Peptidomimetic Vinyl Ester as Falcipain-2 Inhibitors
2012 R. Ettari, N. Micale, G. Grazioso, F. Bova, T. Schirmeister, S. Grasso, M. Zappalà
Mechanism of falcipain-2 inhibition by α,β-unsaturated benzo[1,4]diazepin-2-one methyl ester
2012 G. Grazioso, L. Legnani, L. Toma, R. Ettari, N. Micale, C. De Micheli
Synthesis and anti-HIV activity evaluation of new phenyl ethyl thiourea (PET) derivatives
2009 R. Ettari, A. Pinto, N. Micale