Sfoglia per Autore
Effects of pH and low density lipoprotein (LDL) on PCSK9-dependent LDL receptor regulation
2007 T.S. Fisher, P.L. Surdo, S. Pandit, M. Mattu, J.C. Santoro, D. Wisniewski, R.T. Cummings, A. Calzetta, R.M. Cubbon, P.A. Fischer, A. Tarachandani, R. De Francesco, S.D. Wright, C.P. Sparrow, A. Carfi, A. Sitlani
Advances in the development of new therapeutic agents targeting the NS3-4A serine protease or the NS5B RNA-dependent RNA polymerase of the hepatitis C virus
2007 R. De Francesco, A. Carfí
Phosphorylation of hepatitis C virus NS5A nonstructural protein: A new paradigm for phosphorylation-dependent viral RNA replication?
2007 Y. Huang, K. Staschke, R. De Francesco, S. Tan
Unraveling the hidden catalytic activity of vertebrate class IIa histone deacetylases
2007 A. Lahm, C. Paolini, M. Pallaoro, M.C. Nardi, P. Jones, P. Neddermann, S. Sambucini, M.J. Bottomley, P. Lo Surdo, A. Carfí, U. Koch, R. De Francesco, C. Steinkühler, P. Gallinari
Inhibition of class I histone deacetylase with an apicidin derivative prevents cardiac hypertrophy and failure
2008 P. Gallo, M.V.G. Latronico, P. Gallo, S. Grimaldi, F. Borgia, M. Todaro, P. Jones, P. Gallinari, R. De Francesco, G. Ciliberto, C. Steinkühler, G. Esposito, G. Condorelli
Ezrin is a specific and direct target of protein tyrosine phosphatase PRL-3
2008 E. Forte, L. Orsatti, F. Talamo, G. Barbato, R. De Francesco, L. Tomei
Probing the elusive catalytic activity of vertebrate class IIa histone deacetylases
2008 P. Jones, S. Altamura, R. De Francesco, P. Gallinari, A. Lahm, P. Neddermann, M. Rowley, S. Serafini, C. Steinkühler
A novel series of potent and selective ketone histone deacetylase inhibitors with antitumor activity in vivo
2008 P. Jones, S. Altamura, R. De Francesco, O.G. Paz, O. Kinzel, G. Mesiti, E. Monteagudo, G. Pescatore, M. Rowley, M. Verdirame, C. Steinkühler
Structural and functional analysis of the human HDAC4 catalytic domain reveals a regulatory structural zinc-binding domain
2008 M.J. Bottomley, P.L. Lo Surdo, P.D. Di Giovine, A. Cirillo, R. Scarpelli, F. Ferrigno, P. Jones, P. Neddermann, R. De Francesco, C. Steinkühler, P. Gallinari, A. Carfí
Development and optimization of a binding assay for histone deacetylase 4 using surface plasmon resonance
2008 M. Mattu, P. Di Giovine, C. Steinkuhler, R. De Francesco, S. Altamura, O. Cecchetti, A. Carfì, G. Barbato
Structural and biochemical characterization of the wild type PCSK9-EGF(AB) complex and natural familial hypercholesterolemia mutants
2009 M.J. Bottomley, A. Cirillo, L. Orsatti, L. Ruggeri, T.S. Fisher, J.C. Santoro, R.T. Cummings, R.M. Cubbon, P.L. Surdo, A. Calzetta, A. Noto, J. Baysarowich, M. Mattu, F. Talamo, R. De Francesco, C.P. Sparrow, A. Sitlani, A. Carfí
Naturally occurring hepatitis C virus subgenomic deletion mutants replicate efficiently in Huh-7 cells and are trans-packaged in vitro to generate infectious defective particles
2009 L. Pacini, R. Graziani, L. Bartholomew, R. De Francesco, G. Paonessa
Synthesis and SAR of piperazinyl-N-phenylbenzamides as inhibitors of hepatitis C virus RNA replication in cell culture
2009 I. Conte, C. Giuliano, C. Ercolani, F. Narjes, U. Koch, M. Rowley, S. Altamura, R.D. Francesco, P. Neddermann, G. Migliaccio, I. Stansfield
Loss of histone deacetylase 4 causes segregation defects during mitosis of p53-deficient human tumor cells
2009 B. Cadot, M. Brunetti, S. Coppari, S. Fedeli, E. De Rinaldis, C. Dello Russo, P. Gallinari, R. De Francesco, C. Steinkühler, G. Filocamo
Identification and biological evaluation of a series of 1H-benzo[de]isoquinoline-1,3(2H)-diones as hepatitis C virus NS5B polymerase inhibitors
2009 J.M. Ontoria, E.H. Rydberg, S. Di Marco, L. Tomei, B. Attenni, S. Malancona, J.I. Martin Hernando, N. Gennari, U. Koch, F. Narjes, M. Rowley, V. Summa, S.S. Carroll, D.B. Olsen, R. De Francesco, S. Altamura, G. Migliaccio, A. Carfì
Binding of a Noncovalent Inhibitor Exploiting the S′ region Stabilizes the Hepatitis C virus NS3 Protease Conformation in the Absence of Cofactor
2009 M. Gallo, M. Pennestri, M.J. Bottomley, G. Barbato, T. Eliseo, M. Paci, F. Narjes, R. De Francesco, V. Summa, U. Koch, R. Bazzo, D.O. Cicero
Structural Basis for Resistance of the Genotype 2b Hepatitis C Virus NS5B Polymerase to Site A Non-Nucleoside Inhibitors
2009 E.H. Rydberg, A. Cellucci, L. Bartholomew, M. Mattu, G. Barbato, S.W. Ludmerer, D.J. Graham, S. Altamura, G. Paonessa, R. De Francesco, G. Migliaccio, A. Carfí
Mechanism of hepatitis C virus RNA polymerase inhibition with dihydroxypyrimidines
2010 M.H. Powdrill, J. Deval, F. Narjes, R. De Francesco, M. Götte
Discovery of (7R)-14-Cyclohexyl-7-{[2-(dimethylamino)ethyl](methyl) amino}-7,8-dihydro-6H-indolo[1,2-e][1,5]benzoxazocine-11-carboxylic Acid (MK-3281), a Potent and Orally Bioavailable Finger-Loop Inhibitor of the Hepatitis C Virus NS5B Polymerase
2011 F. Narjes, B. Crescenzi, M. Ferrara, J. Habermann, S. Colarusso, M. Del Rosario Rico Ferreira, I. Stansfield, A.C. Mackay, I. Conte, C. Ercolani, S. Zaramella, M. Palumbi, P. Meuleman, G. Leroux-Roels, C. Giuliano, F. Fiore, S. Di Marco, P. Baiocco, U. Koch, G. Migliaccio, S. Altamura, R. Laufer, R. De Francesco, M. Rowley
Distinct microRNA signatures in human lymphocyte subsets and enforcement of the naive state in CD4+ T cells by the microRNA miR-125b
2011 R.L. Rossi, G. Rossetti, L. Wenandy, S. Curti, A. Ripamonti, R.J.P. Bonnal, R.S. Birolo, M. Moro, M.C. Crosti, P. Gruarin, S. Maglie, F. Marabita, D. Mascheroni, V. Parente, M. Comelli, E. Trabucchi, R. De Francesco, J. Geginat, S. Abrignani, M. Pagani
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