Sfoglia per Autore
4-Aminoquinoline quinolizidinyl- and quinolizidinylalkyl-derivatives with antimalarial activity
2005 A. Sparatore, N. Basilico, S. Parapini, S. Romeo, F. Novelli, F. Sparatore, D. Taramelli
Design and synthesis of novel antimalarial agents based on a polyaromatic scaffold
2006 G. Campiani, S. Gemma, C. Fattorusso, M. Persico, S. Butini, G. Kukreja, B.P. Joshi, E. Fattorusso, D. Taramelli, N. Basilico, V. Yardley
Effetti antiangiogenetici di derivati di artemisinina, una classe di composti ad attività antimalarica e antitumorale
2006 S. D'Alessandro, M. Gelati, N. Basilico, R. Haynes, D. Taramelli
Antimalarial activity of novel pyrrolizidinyl derivatives of 4-aminoquinolines
2006 A. Sparatore, S. Romeo, N. Basilico, S. Parapini, D. Taramelli, S. Wittlin, R. Brun, F. Sparatore
Design, synthesis, and in vitro biological evaluation of 7-chloro-4-quinolylhydrazones as promising anti-malarial agents
2006 S. Butini, S. Gemma, C. Fattorusso, M. Persico, G. Kukreja, P.J. Bhupendra, E. Fattorusso, D. Taramelli, N. Basilico, V. Yardley, G. Campiani, V. Nacci
Inhibition of angiogenesis and of erythroid differentiation by artemisinin derivatives
2006 S. D'Alessandro, M. Gelati, N. Basilico, R.K. Haynes, D. Taramelli
In vivo activity of quinolizidinyl-and quinolizidynilalkyl-derivatives of 4-aminoquinoline on the murine malaria parasite Plasmodium berghei
2006 L. Lucantoni, A. Sparatore, B. Barbosa, N. Basilico, S. Parapini, V. Yardley, L. Stewart, A. Habluetzel, L. Pasqualini, F. Esposito, D. Taramelli
In vivo evaluation of quinolizidinyl-and quinolizidinylalkyl-derivatives of 4-aminoquinoline using the murine malaria model Plasmodium berghei/anopheles stephensi
2006 L. Lucantoni, A. Sparatore, N. Basilico, S. Parapini, V. Yardley, L. Stewart, A. Habluetzel, L. Pasqualini, F. Esposito, D. Taramelli
Haem metabolism in Plasmodium falciparum : consequences for the parasites and host cells
2006 D. Taramelli, N. Basilico, S. Parapini, D. Monti
Endoperoxide derivatives from marine organisms: 1,2-dioxanes of the plakortin family as novel antimalarial agents
2006 C. Fattorusso, G. Campiani, B. Catalanotti, M. Persico, N. Basilico, S. Parapini, D. Taramelli, C. Campagnuolo, E. Fattorusso, A. Romano, O. Taglialatela-Scafati
Synthesis of N1-arylidene-N2-quinolyl- and N2-acrydinylhydrazones as potent antimalarial agents activa against CQ-resistant P. falciparum strains
2006 S. Gemma, G. Kukreja, C. Fattoruso, M. Persico, M.P. Romano, M. Altarelli, L. Savini, G. Campiani, E. Fattorusso, N. Basilico, D. Taramelli, V. Yardley, S. Butini
Insights on the mechanism of action of novel quinolizidinyl-and quinolizidinylalkyl-derivatives with antimalarial activity
2006 S. Parapini, A. Sparatore, T.J. Egan, N. Basilico, B. Barbosa, S. Romeo, D. Jabès, D. Taramelli
Design and synthesis of potent antimalarial agents based on clotrimazole scaffold : exploring an innovative pharmacophore
2007 S. Gemma, G. Campiani, S. Butini, G. Kukreja, B.P. Joshi, M. Persico, B. Catalanotti, E. Novellino, E. Fattorusso, V. Nacci, L. Savini, D. Taramelli, N. Basilico, G. Morace, V. Yardley, C. Fattorusso
Combined effects of artemisinin and quinoline derivatives on mammalian cell growth and differentiation
2007 S. Finaurini, N. Basilico, S. D’Alessandro, D. Monti, S.A. Ward, D. Taramelli
Effects of artemisinin and quinoline derivatives on K562 cell differentiation
2007 S. Finaurini, N. Basilico, S. D’Alessandro, D. Monti, S.A. Ward, D. Taramelli
Development of piperazine-tethered heterodimers as potent antimalarials against chloroquine-resistant P.falciparum strains : synthesis and molecular modeling
2007 S. Gemma, G. Kukreja, G. Campiani, S. Butini, M. Bernetti, B.P. Joshi, L. Savini, N. Basilico, D. Taramelli, V. Yardley, A. Bertamino, E. Novellino, M. Persico, B. Catalanotti, C. Fattorusso
Differential effects on angiogenesis of two antimalarial compounds, dihydroartemisinin and artemisone : implications for embryotoxicity
2007 S. D'Alessandro, M. Gelati, N. Basilico, E.A. Parati, R.K. Haynes, D. Taramelli
Novel 4-aminoquinolines through microwave-assisted SNAr reactions : a practical route to antimalarial agents
2007 S. Melato, P. Coghi, N. Basilico, D. Prosperi, D. Monti
Old and new targets for innovative antimalarial compounds : the different strategies of the Italian Malaria Network
2008 N. Basilico, E. Bosisio, F. Buelli, G. Campiani, M. Casagrande, F. Castelli, P. Coghi, Y. Corbett, L. Cortelezzi, S. D'Alessandro, M. Dell'Agli, F. Esposito, C. Fattorusso, E. Fattorusso, S. Finaurini, G.V. Galli, S. Gemma, A. Habluetzel, L. Lucantoni, S.R. Melato, D. Monti, P. Olliaro, M.F. Omodeo-Salè, S. Parapini, M. Persico, M. Rizzi, S. Romeo, F. Rossi, C. Rusconi, A. Sparatore, O.T. Scafati, E. van den Bogaart, D. Taramelli, N. Vaiana, S. Yerbanga
Anti-plasmodial activity of Ailanthus excelsa
2008 M. Dell'Agli, G. Galli, S. Parapini, N. Basilico, D. Taramelli, A. Said, K. Rashed, E.A. Bosisio
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