(αR,2R)- and (αR,2S)-2-methyl-4-(α-phenylethyl)-1,2,3,4- tetrahydro-benzo[e][1,4]diazepin-5-ones 7 and 8 were synthesised by an intramolecular azide cycloaddition followed by stereoselective reduction of a bicyclic ketimine.
Diastereoselective synthesis of enantiopure (aR)-2-methyl-4-(a-phenylethyl)-1,2,3,4-tetrahydro-benzo[e][1,4]diazepin-5-ones / E.M. Beccalli, G. Broggini, G. Paladino, T. Pilati, G. Pontremoli. - In: TETRAHEDRON-ASYMMETRY. - ISSN 0957-4166. - 15:4(2004), pp. 687-692. [10.1016/j.tetasy.2003.11.033]
Diastereoselective synthesis of enantiopure (aR)-2-methyl-4-(a-phenylethyl)-1,2,3,4-tetrahydro-benzo[e][1,4]diazepin-5-ones
E.M. BeccalliPrimo
;
2004
Abstract
(αR,2R)- and (αR,2S)-2-methyl-4-(α-phenylethyl)-1,2,3,4- tetrahydro-benzo[e][1,4]diazepin-5-ones 7 and 8 were synthesised by an intramolecular azide cycloaddition followed by stereoselective reduction of a bicyclic ketimine.
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