MASCIOCCHI, DANIELA
MASCIOCCHI, DANIELA
Dipartimento di Scienze Farmaceutiche
An in vivo active 1,2,5-oxadiazole Pt(II) complex : a promising anticancer agent endowed with STAT3 inhibitory properties
2017 F. Porta, G. Facchetti, N. Ferri, A. Gelain, F. Meneghetti, S. Villa, D. Barlocco, D. Masciocchi, A. Asai, N. Miyoshi, S. Marchianò, B. Kwon, Y. Jin, V. Gandin, C. Marzano, I. Rimoldi
Ureido-pyridazinone derivatives : insights into the structural and conformational properties for STAT3 inhibition
2015 F. Meneghetti, S. Villa, D. Masciocchi, D. Barlocco, L. Toma, D-C. Han, B-M. Kwon, N. Ogo, A. Asai, L. Legnani, A. Gelain
Modeling, synthesis and NMR characterization of novel chimera compounds targeting STAT3
2014 S. Dell'Orto, D. Masciocchi, S. Villa, F. Meneghetti, G. Celentano, D. Barlocco, D. Colombo, L. Legnani, L.A. Toma, Y.J. Jeon, B. Kwon, A. Asai, A. Gelain
Crystal structure of 3-(3-oxo-2,3,4,4a,5,6-hexahydrobenzo[h]cinnolin-2-yl)propionic acid
2014 F. Meneghetti, D. Masciocchi, A. Gelain, S. Villa
Sviluppo di MD77: nuovi derivati eterociclici inibenti STAT3
2014 A. Gelain, F. Porta, S. Dell’Orto, S. Villa, D. Masciocchi, D. Barlocco, F. Meneghetti, N. Ferri, G. Poli, T. Tuccinardi, B.M. Kwon, A. Asai
Synthesis, structure-activity relationships and stereochemical investigations on new tricyclic pyridazinone derivatives as potential STAT3 inhibitors
2013 F. Meneghetti, D. Masciocchi, A. Gelain, F. Porta, A. Pedretti, G. Celentano, D. Barlocco, L. Legnani, L. Toma, B. Kwon, A. Asai, S. Villa
Synthesis, structure–activity relationships andstereochemical investigations of new tricyclic pyridazinone derivatives as potential STAT3 inhibitors
2013 D. Masciocchi, A. Gelain, F. Porta, F. Meneghetti, A. Pedretti, G. Celentano, D. Barlocco, L. Legnani, L. Toma, B.M. Kwon, A. Asai, S. Villa
Identification of a novel STAT3 inhibitor structurally related to the oxadiazole derivative MD77
2013 D. Masciocchi, S. Villa, F. Porta, D. Barlocco, F. Meneghetti, B.M. Kwon, A. Asai, A. Gelain
Exploring scaffolds to discover new STAT3 inhibitors, as novel anticancer agents.
2012 S. Villa, D. Masciocchi, A. Gelain, S. Dell'Orto, F. Meneghetti, A. Pedretti, D. Barlocco, L. Legnani, L. Yoma, B._.M. Kwon, S. Nakano, A. Asai
Optimation of the lead MD77
2012 D. Barlocco, S. Villa, D. Masciocchi, A. Gelain, F. Meneghetti, B. Kwon
DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF POTENTIAL STAT3 INHIBITORS AS ANTICANCER AGENTS
2012 D. Masciocchi
New STAT3 inhibitors: identification of a lead
2012 A. Gelain, D. Masciocchi, S. Villa, F. Meneghetti, A. Pedretti, D. Barlocco, L. Legnani, L. Toma, B.M. Kwon, S. Nakano, A. Asai
Merged structures as new STAT3 inhibitors: the chimera compounds
2012 A. Gelain, D. Masciocchi, S. Villa, S. Dell’Orto, F. Meneghetti, A. Pedretti, D. Barlocco, L. Legnani, L. Toma, B. Kwon, S. Nakano, A. Asai
The influence of the substitution pattern on the molecular conformation of ureido 1,2,5-oxadiazoles, related to STAT3 inhibitors: chemical behavior and structural investigation
2012 S. Villa, D. Masciocchi, A. Gelain, F. Meneghetti
Chemical behaviour and crystallographic characterization of ureido 1,2,5-oxadiazole derivatives, related to Stat3 inhibitors
2011 F. Meneghetti, D. Masciocchi, A. Gelain, S. Villa
Signal transducer and activator of transcription (Stat) 3: a promising target for anticancer therapy
2011 D. Masciocchi, A. Gelain, S. Villa, F. Meneghetti, D. Barlocco
Synthesis, modeling, and crystallographic study of 3,4-disubstituted-1,2,5-oxadiazoles and evaluation of their ability to decrease STAT3 activity
2010 D.S. Shin, D. Masciocchi, A. Gelain, S. Villa, D. Barlocco, F. Meneghetti, A. Pedretti, Y.M. Han, D.C. Han, M.Y. Han, B.M. Kwon, L. Legnani, L. Toma
Tricyclic Pyridazinone derivatives : development of new STAT-3 inhibitors
2010 A. Gelain, D. Masciocchi, S. Villa, A. Pedretti, F. Meneghetti, D. Barlocco, B.M. Kwon, D.S. Shin, L. Legnani, L. Toma
Development on furazan derivatives as potential STAT-3 inhibitors
2009 D. Masciocchi, S. Villa, A. Gelain, A. Pedrettti, F. Meneghetti, D. Barlocco, B.M. Kwon, A. Pedretti
Studies on potential STAT-3 inhibitors: reactivity and behaviour of furazan derivatives
2009 D. Masciocchi, S. Villa, A. Gelain, F. Meneghetti, A. Pedretti, D. Barlocco, B.M. Kwon