2-Thiazolin-4-one derivatives, obtained by reaction of tert-butyl (3-methoxy-1-methyl-3-oxoprop-1-enyl)diazenecarboxylate with aryl thioamides, were transformed into 5-bromoacetyl-4-hydroxythiazole derivatives by polymer-supported reagents and simple work-up procedures. The compounds thus synthesised were coupled with thioamides bearing valuable functional groups affording novel polyfunctionalised 4,5′-bithiazol-4′-ol derivatives
Efficient synthesis of novel polyfunctionalised 4,5’-bithiazol-4’-ol derivatives / A. Arcadi, O.A. Attanasi, P. Filippone, F.R. Perulli, E. Rossi, S. Santeusanio. - In: SYNLETT. - ISSN 0936-5214. - 2004:15(2004), pp. 2681-2684.
Efficient synthesis of novel polyfunctionalised 4,5’-bithiazol-4’-ol derivatives
E. RossiPenultimo
;
2004
Abstract
2-Thiazolin-4-one derivatives, obtained by reaction of tert-butyl (3-methoxy-1-methyl-3-oxoprop-1-enyl)diazenecarboxylate with aryl thioamides, were transformed into 5-bromoacetyl-4-hydroxythiazole derivatives by polymer-supported reagents and simple work-up procedures. The compounds thus synthesised were coupled with thioamides bearing valuable functional groups affording novel polyfunctionalised 4,5′-bithiazol-4′-ol derivatives
Pubblicazioni consigliate
I documenti in IRIS sono protetti da copyright e tutti i diritti sono riservati, salvo diversa indicazione.
