Sfoglia per Autore
Tricyclic 3-(2H)-pyridazinone derivatives : synthesis and evaluation of their antisecretory and antiulcer activity
1992 G. Cignarella, D. Barlocco, S. Villa, M. Curzu, G. Pinna, A. Lavezzo, A. Bestetti
Synthesis of a new series of 8-substituted-2,8-diazaspiro(4,5)decan-3-ones
1993 G. Cignarella, S. Villa, D. Barlocco
Synthesis and pharmacological evaluation of a new class of 2-oxo-8-azaspiro(4,5)decan-1-ones as analogues of the muscarinic agonist RS-86
1993 G. Cignarella, S. Villa, D. Barlocco
Synthesis of a new series of N-substituted-3(1-alkyl/aryl-4-piperidyl)azetidin-2-ones as possible muscarinic agents
1993 G. Cignarella, S. Villa, D. Barlocco
Synthesis of a new series of 2.8-disubstituted-2,8-diazaspiro(4,5)decan-1-ones as potential muscarinic agonists
1994 G. Cignarella, S. Villa, F. Cattabeni, F. Renò, M. Cimino, P.G. De benedetti, D. Barlocco
Synthesis of a new series of 2,7-diazaspiro(3,5)nonan-1-ones and study of their cholinergic properties
1994 G. Cignarella, S. Villa, D. Barlocco
MONOCYCLIC ANALOGS OF THE MU-OPIOID AGONIST 3,8-DIAZABICYCLO-[3.2.1]OCTANES - SYNTHESIS, MODELING, AND ACTIVITY
1995 D. BARLOCCO, S. VILLA, W. FRATTA, P. FADDA, D. COLOMBO, L. TOMA
2-(Substituted)amino-2,8-diazaspiro[4,5]decan-1,3-diones as potential muscarinic agonists: Synthesis, modeling and binding studies
1996 D. Barlocco, F. Fanelli, G. Cignarella, S. Villa, F. Cattabeni, W. Balduini, M. Cimino, P.G. De Benedetti
Valutazione in vivo di molecole applicabili alla terapia delle encefalopatie spongiformi trasmissibili
1997 S. Russo, B. Canciani, M. Porro, S. Villa, A. Cocilovo, G. Cignarella, P. Mantegazza, F. Tagliavini, G. Poli
Benzocondensed derivatives as rigid analogues of the -opioid agonist 3(8)-cinnamyl-8(3)-propionyl-3,8-diazabicyclo[3.2.1]octanes: synthesis, modeling, and affinity
1998 G. Cignarella, D. Barlocco, P. Vianello, S. Villa, G.A. Pinna, P. Fadda, W. Fratta, L. Toma, S. Gessi
Mono- and disubstituted-3,8-diazabicyclo[3.2.1]octane derivatives as analgesics structurally related to epibatidine: Synthesis, activity, and modeling
1998 D. Barlocco, G. Cignarella, D. Tondi, P. Vianello, S. Villa, A. Bartolini, C. Ghelardini, N. Galeotti, D. Anderson, T. Kuntzweiler, D. Colombo, L. Toma
Synthesis and mu-opioid receptor affinity of a new series of nitro substituted 3,8-diazabicyclo[3.2.1]octane derivatives
1998 D. Barlocco, G. Cignarella, P. Vianello, S. Villa, G.A. Pinna, P. Fadda, W. Fratta
Pyridazinones and their tricyclic congeners : chemistry and biology
1998 G. Cignarella, D. Barlocco, S. Villa, M.M. Curzu, G.A. Pinna
Valutazione in vivo delle potenzialità terapeutiche di nuove molecole nel trattamento delle encefalopatie spongiformi trasmissibili
1998 G. Carcassola, P. Dall'Ara, S. Russo, F. Tagliavini, G. Cignarella, S. Villa
Behaviour of 5,6-dihydrothieno[2,3-h]cinnolin-3(2H)-one and 5,6-dihydrothieno[3,2-h]cinnolin-3(2H)-one towards hydrazine. Synthesis of thienocinnolinones and of 4-aminothienocinnolinones
1999 S. Villa, G. Cignarella, M.M. Curzu, G.A. Pinna, E. Pini, L. Toma
Behavior of 5,6-dihydrobenzo[h]cinnolinones towards hydrazine. Synthesis of benzo[h]cinnolinones and of 4-aminobenzo[h]cinnolinones
1999 S. Villa, G.L. Evoli, G. Cignarella, M.M. Curzu, G.A. Pinna
Synthesis, modelling, and mu-opioid receptor affinity of N-3(9)-arylpropenyl-N-9(3)-propionyl-3,9-diazabicyclo[3.3.1]nonanes
2000 G. Pinna, G. Murineddu, M. Curzu, S. Villa, P. Vianello, P. Borea, S. Gessi, L. Toma, D. Colombo, G. Cignarella
3,8-diazabicyclo[3.2.1]octane derivatives as analogues of abasilide, a class III antiarrhythmic agent
2001 S. Villa, D. Barlocco, G. Cignarella, G.J. Papp, B. Balati, J. Takacs, A. Varrò, K. Keseru, P. Matyus
Determination of sodium 3,4-diaminonaphtalene-1-sulfonate, a Congo Red derivative, in plasma and brain of hamsters by high-performance liquid chromatography after solid-phase extraction and ultraviolet absorbance
2002 R. Pirola, M. Gervasoni, C. Pollera, S. Villa, P. Mantegazza, S.R. Bareggi
Congo red analogues as potential anti-prion agents
2003 S. Villa, G. Cignarella, D. Barlocco, M. Gervasoni, G. Carcassola, L. Giannino, P. Mantegazza
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