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Mostrati risultati da 1 a 20 di 27
Titolo Data di pubblicazione Autori Tipo File Abstract
Oxidation State Dependent Conformational Changes of HMGB1 Regulate the Formation of the CXCL12/HMGB1 Heterocomplex 2019 Fassi E. M. A.Grazioso G. + Article (author) -
Exploring Proprotein Convertase Subtilisin/Kexin 9 (PCSK9) Autoproteolysis Process by Molecular Simulations: Hints for Drug Design 2020 Fassi, Enrico M ALammi, CarmenRoda, GabriellaGrazioso, Giovanni + Article (author) -
Trans-Epithelial Transport, Metabolism and Biological Activity Assessment of the Multi-Target Lupin Peptide LILPKHSDAD (P5) and Its Metabolite LPKHSDAD (P5-Met) 2021 C. LammiC. BollatiJ. LiM. BartolomeiE. M. A. FassiG. GraziosoA. Arnoldi + Article (author) -
Structure, Immunoreactivity, and In Silico Epitope Determination of {SmSPI} S. mansoni Serpin for Immunodiagnostic Application 2021 Stefano De BenedettiFlavio Di PisaEnrico Mario Alessandro FassiMartino BolognesiMaria Rita GismondoDavide MiletoAlessandro ManconLouise Jane Gourlay + Article (author) -
Investigation of Chlorella pyrenoidosa Protein as a Source of Novel Angiotensin I-Converting Enzyme (ACE) and Dipeptidyl Peptidase-IV (DPP-IV) Inhibitory Peptides 2021 Y. LiE. M. A. FassiG. BoschinM. BartolomeiC. BollatiG. RodaA. ArnoldiG. GraziosoC. Lammi + Article (author) -
Systematic Development of Peptide Inhibitors Targeting the CXCL12/HMGB1 Interaction 2021 Fassi E. M. A.Grazioso G. + Article (author) -
Analysis of Hsp90 allosteric modulators interactome reveals a potential dual action mode involving mitochondrial MDH2 2021 Fassi E. M. A.Sattin S. + Article (author) -
Elucidating the 3D Structure of a Surface Membrane Antigen from Trypanosoma cruzi as a Serodiagnostic Biomarker of Chagas Disease 2022 Di Pisa F.De Benedetti S.Fassi E. M. A.Mileto D.Mancon A.Gori A.Bolognesi M.Gourlay L. J. + Article (author) -
Computational Design and Biological Evaluation of Analogs of Lupin Peptide P5 Endowed with Dual PCSK9/HMG-CoAR Inhibiting Activity 2022 C. LammiE. FassiJ. LiM. BartolomeiG. RodaA. ArnoldiG. Grazioso + Article (author) -
Focused Design of Novel Cyclic Peptides Endowed with GABARAP-Inhibiting Activity 2022 Enrico Mario Alessandro FassiMichele Dei CasMatteo MoriGabriella RodaGiovanni Grazioso + Article (author) -
Natural compounds targeting E. Coli WRBA as antibiofilm agents: Virtual screening, design and synthesis of analogs, biological evaluation 2022 Villa, S.Mori, M.Meneghetti, F.Roda, G.Gelain, A.Villa F.Fassi, E.Forlani,F.Grazioso, G + Conference Object -
Elagolix analogues as potential new GnRH antagonists 2022 Ciceri SamueleColombo DiegoFassi EnricoFerraboschi PatriziaGrazioso GiovanniMeneghetti Fiorella + Conference Object -
Elagolix analogues as potential new GnRH antagonists: design, synthesis and characterization 2022 Ciceri SamueleColombo DiegoFassi EnricoFerraboschi PatriziaGrazioso GiovanniMeneghetti Fiorella + Conference Object -
Computational Design, Synthesis, and Biological Evaluation of Diimidazole Analogues Endowed with Dual PCSK9/HMG-CoAR-Inhibiting Activity 2023 Carmen LammiEnrico M. A. FassiMarco ManentiJianqiang LiGabriella RodaMarina CameraAlessandra SilvaniGiovanni Grazioso + Article (author) -
Mechanistic Insights into the Antibiofilm Mode of Action of Ellagic Acid 2023 Ratti, AlessandroFassi, Enrico M. A.Forlani, FabioMori, MatteoVilla, FedericaCappitelli, FrancescaRoda, GabriellaVilla, StefaniaGrazioso, Giovanni + Article (author) -
Unlocking the Antibiofilm Potential of Natural Compounds by Targeting the NADH:quinone Oxidoreductase WrbA 2023 Alessandro RattiEnrico M. A. FassiFabio ForlaniMaurizio ZangrossiMatteo MoriFrancesca CappitelliGabriella RodaStefania VillaFederica VillaGiovanni Grazioso Article (author) -
Elagolix Sodium Salt and Its Synthetic Intermediates: A Spectroscopic, Crystallographic, and Conformational Study 2023 Samuele CiceriDiego ColomboEnrico M. A. FassiPatrizia FerraboschiGiovanni GraziosoCarlo CastellanoFiorella Meneghetti + Article (author) -
Computational Design, Synthesis, and Biophysical Evaluation of β-Amido Boronic Acids as SARS-CoV-2 Mpro Inhibitors 2023 Fassi, Enrico M. A.Manenti, MarcoCitarella, AndreaDei Cas, MicheleCasati, SaraRoda, GabriellaSilvani, AlessandraGrazioso, Giovanni + Article (author) -
Development of AMBER Parameters for Molecular Simulations of Selected Boron-Based Covalent Ligands 2023 Fassi, Enrico Mario AlessandroRoda, GabriellaGrazioso, Giovanni + Article (author) -
COMPUTATIONAL DESIGN OF PEPTIDES AND PEPTIDOMIMETICS AS POTENTIAL THERAPEUTIC AGENTS TO SATISFY PRESSING MEDICAL NEEDS 2023 FASSI, ENRICO MARIO ALESSANDRO Doctoral Thesis -
Mostrati risultati da 1 a 20 di 27
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