Sfoglia per Autore
ANALOGHI STRUTTURALI DEL WB 4101: PROGETTAZIONE, SINTESI E VALUTAZIONE BIOLOGICA
2004 C. Bolchi, L. Fumagalli, B. Moroni, M. Pallavicini, C.M. Rusconi, E. Valoti
Univocal syntheses of 2- and 3-hydroxymethyl-2,3-dihydro[1,4]dioxino[2,3-b]pyridine enantiomers
2005 C. Bolchi, M. Pallavicini, L. Fumagalli, B. Moroni, C. Rusconi, E. Valoti
Highly efficient resolutions of 1,4-benzodioxane-2-carboxylic acid with para substituted 1-phenylethylamines
2005 C. Bolchi, M. Pallavicini, L. Fumagalli, N. Marchini, B. Moroni, C. Rusconi, E. Valoti
ANALOGUES OF ALPHA1-ADRENOCEPTOR ANTAGONIST WB4101: DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION
2005 C. Bolchi, R. Budriesi, A. Chiarini, L. Fumagalli, M. Gobbi, P. Ioan, B. Moroni, M. Pallavicini, C. Rusconi, E. Valoti
SEARCH FOR SELECTIVE ANTAGONISTS AT α1-ADRENORECEPTOR SUBTYPES: WB-4101 RELATED COMPOUNDS
2005 C. Bolchi, R. Budriesi, A. Chiarini, L. Fumagalli, M. Gobbi, P. Ioan, B. Moroni, M. Pallavicini, C.M. Rusconi, E. Valoti
Synthesis and a4b2 nicotinic affinity of the stereoisomers of 2-(1-methyl-2-pyrrolidinyl)-1,4-benzodioxane and of its nor-methyl derivative
2007 C. Bolchi, A. Cilia, R. Ferrara, L. Fumagalli, A. Gaimarri, C. Gotti, M. Pallavicini, C.M. Rusconi, E. Valoti
Resolution of 2-substituted 1,4-benzodioxanes by entrainment
2007 C. Bolchi, M. Pallavicini, L. Fumagalli, C. Rusconi, M. Binda, E. Valoti
Peptidomimetic inhibitors of farnesyltransferase with high in vitro activity and significant cellular potency
2007 C. Bolchi, M. Pallavicini, C. Rusconi, L. Diomede, N. Ferri, A. Corsini, L. Fumagalli, A. Pedretti, G. Vistoli, E. Valoti
Old and new targets for innovative antimalarial compounds : the different strategies of the Italian Malaria Network
2008 N. Basilico, E. Bosisio, F. Buelli, G. Campiani, M. Casagrande, F. Castelli, P. Coghi, Y. Corbett, L. Cortelezzi, S. D'Alessandro, M. Dell'Agli, F. Esposito, C. Fattorusso, E. Fattorusso, S. Finaurini, G.V. Galli, S. Gemma, A. Habluetzel, L. Lucantoni, S.R. Melato, D. Monti, P. Olliaro, M.F. Omodeo-Salè, S. Parapini, M. Persico, M. Rizzi, S. Romeo, F. Rossi, C. Rusconi, A. Sparatore, O.T. Scafati, E. van den Bogaart, D. Taramelli, N. Vaiana, S. Yerbanga
In vitro and in vivo evaluation and early transitioning studies of novel quinolizidinyl- and quinolizidinylalkyl- derivatives of 4-aminoquinoline with potent antimalarial activity
2008 D. Taramelli, N. Basilico, M. Casagrande, Y. Corbett, S. Parapini, S. Romeo, C. Rusconi, A. Tosi, L. Vivas, E. van den Bogaart, D. Jabes, A. Sparatore
New Ras CAAX mimetics : design, synthesis, antiproliferative activity, and RAS prenylation inhibition
2009 C. Bolchi, M. Pallavicini, L. Fumagalli, N. Ferri, A. Corsini, C. Rusconi, E. Valoti
Antiparasitic activities and toxicities of individual enantiomers of 7-chloro-N-[[(9a)-octahydro-2H-quinolizin-1-yl]methyl]-4-quinolinamine
2009 D. Taramelli, A. Sparatore, S. Romeo, N. Basilico, N. Vaiana, M. Casagrande, L. Rizzi, S. D’Alessandro, S. Parapini, C. Rusconi, H. Lander, L. Vivas, D. Jabes
Antiparasitic activity and ADME-Tox profile of new 4-aminoquinoline derivatives
2010 C. Rusconi, M. Casagrande, N. Basilico, V. Tazzari, N. Vaiana, L. Vivas, S. Romeo, D. Taramelli, A. Sparatore
Novel arylpyrrolylaminoquinolines as potent antimalarial agents
2010 M. Casagrande, C. Rusconi, N. Basilico, D. Taramelli, A. Sparatore
Antiparasitic activity and ADME-tox profile of new 4-aminoquinoline derivatives
2010 C. Rusconi, A. Sparatore, N. Basilico, S. Romeo, N. Vaiana, M. Casagrande, L. Rizzi, V. Tazzari, L. Vivas, P. Verducci, D. Jabes, D. Taramelli
NOVEL ARYLPYRROLYLAMINOQUINOLINES AS POTENT ANTIMALARIAL AGENTS
2010 M. Casagrande, C. Rusconi, N. Basilico, D. Taramelli, A. Sparatore
Synthesis, antimalarial activity, and cellular toxicity of new arylpyrrolylaminoquinolines
2010 M. Casagrande, N. Basilico, C. Rusconi, D. Taramelli, A. Sparatore
How selection was made for a new antimalarial drug candidate : from AM1 to MG3, two novel series of 4-aminoquinoline derivatives
2011 C. Rusconi, M. Casagrande, V. Tazzari, N. Vaiana, Y. Corbett, N. Basilico, L. Cortelezzi, D. Scaccabarozzi, F. Omodeo Salè, S. Romeo, D. Taramelli, A. Sparatore
Scale-up synthesis of MG3, a pyrrolizidinyl 4-aminoquinoline derivative, as novel antimalarial drug candidate
2011 N. Vaiana, C. Rusconi, A. Pancotti, V. Tazzari, A. Sparatore, S. Romeo
Synthesis and antiplasmodial evaluation of new N-(imidazol-2-yl)-methyl-4-aminoquinolines
2011 M. Casagrande, A. Barteselli, C. Rusconi, S. Parapini, D. Ilboudo, D. Taramelli, A. Sparatore
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