Sfoglia per Autore
The impact of Chirality on Medicinal Chemistry
2003 M. De Amici, P. Conti, C. Dallanoce, G. Grazioso, S. Joppolo di Ventimiglia, M. Racca, G. Roda, C. De Micheli
Design of Cyclopentaisoxazoline Amino Acids as Conformationally Constrained Agonists at Glutamate Receptors
2003 P. Conti, M. De Amici, G. Grazioso, G. Roda, T.B. Stensbøl, H. Bräuner-Osborne, U. Madsen, L. Toma, C. De Micheli
Design of Cyclopentaisoxazoline Amino Acids as Conformationally Constrained Agonists at Glutamate Receptors
2003 P. Conti, M. De Amici, G. Grazioso, G. Roda, T.B. Stensbøl, H. Bräuner-Osborne, U. Madsen, L. Toma, C. De Micheli
Design, synthesis, and pharmacological characterization of novel, potent NMDA receptor antagonists
2004 P. Conti, M. De Amici, G. Grazioso, G. Roda, F.F. Barberis Negra, B. Nielsen, T.B. Stensbl, U. Madsen, H. Bräuner Osborne, K. Frydenvang, G. De Sarro, L. Toma, C. De Micheli
Synthesis of Novel N1-Substituted Bicyclic Pyrazole Amino Acids and Evaluation of Their Interaction with Glutamate Receptors
2005 P. Conti, G. Grazioso, S. Joppolo di Ventimiglia, A. Pinto, G. Roda, U. Madsen, H. Bräuner Osborne, B. Nielsen, C. Costagli, A. Galli
Development of a Three-Dimensional Model for the N-Methyl-D-aspartate NR2A Subunit
2005 G. Grazioso, L. Moretti, L. Scapozza, M. De Amici, C. De Micheli
Synthesis and binding affinity at neuronal nicotinic acetylcholine receptors of novel epibatidine-related delta2-isoxazoline derivatives
2005 P. Bazza, C. Dallanoce, G. Grazioso, M. De Amici, C. De Micheli, C. Gotti, L. Riganti, F. Clementi
Synthesis, Binding Affinity at Glutamic Acid Receptors, Neuroprotective Effects, and Molecular Modeling Investigation of Novel Dihydroisoxazole Amino Acids
2005 P. Conti, M. De Amici, G. Grazioso, G. Roda, A. Pinto, K.B. Hansen, B. Nielsen, U. Madsen, H. Brauner Osborne, J. Egebjerg, V. Vestri, D.E. Pellegrini Giampietro, P. Sibille, F.C. Acher, C. De Micheli
Molecular Modeling of New Ligands Selective for the NMDA Receptors
2006 G. Grazioso
Synthesis, chiral resolution, and enantiopharmacology of a potent 2,3-benzodiazepine derivative as noncompetitive AMPA receptor antagonist
2006 M. Zappalà, G. Postorino, N. Micale, S. Caccamese, N. Parrinello, G. Grazioso, G. Roda, F.S. Menniti, G. De Sarro, S. Grasso
Synthesis of novel epibatidine-related derivatives through 1,3-dipolar cycloaddition of pyridinenitrile oxides
2006 C.M.L. Dallanoce, P. Bazza, G. Grazioso, M. De Amici, C. De Micheli
Synthesis of epibatidine-related Delta(2)-isoxazoline derivatives and evaluation of their binding affinity at neuronal nicotinic acetylcholine receptors
2006 C.M.L. Dallanoce, P. Bazza, G. Grazioso, M. De Amici, C. Gotti, L. Riganti, F. Clementi, C. De Micheli
Synthesis of 3-hydroxy- and 3-carboxy-Delta(2)-isoxazoline amino acids and evaluation of their interaction with GABA receptors and transporters
2006 P. Conti, M. De Amici, A. Pinto, L. Tamborini, G. Grazioso, B. Frolund, B. Nielsen, C. Thomsen, B. Ebert, C. De Micheli
Molecular Modeling Investigation of ligands acting as Glucoamylase II inhibitors
2007 J. Sgrignani, C. Bonaccioni, M. Chioccioli, F. Cardona, A. Goti, G. Grazioso, P. Gratteri
Determinazione dell’energia di legame di agonisti del recettore nicotinico alpha-7 mediante applicazione dell’approccio MMPB(GB)SA
2007 G. Grazioso, A. Cavalli, M. Recanatini, M. De Amici, C. De Micheli
Synthesis of novel enantiopure 2-isoxazoline and 2-pyrazoline amino acids and their activity at glutamic acid receptors and transporters
2007 P. Conti, A. Pinto, L. Tamborini, G. Grazioso, G. Roda, M. De Amici, C. DE MICHELI
(-)-HIP-A and (+)-HIP-B: investigation of the pharmacological profile and potential therapeutic applications
2007 P. Conti, A. Pinto, L. Tamborini, G. Grazioso, S. Colleoni, M. Gobbi, T. Mennini
Agonisti nicotinici selettivi nel trattamento di patologie del Sistema Nervoso Centrale
2007 C. De Micheli, M. De Amici, C. Dallanoce, G. Grazioso, L. Rizzi, P. Magrone, C. Matera
Synthesis of Conformationally Constrained Glutamic Acid Homologues and Investigation of Their Pharmacological Profiles
2007 P. Conti, A. Pinto, L. Tamborini, G. Grazioso, G. De Sarro, H. Brauner Osborne, G. Szabo, L.G. Harsing, C. De Micheli
Evaluation of binding free energy of nicotinic agonists by the linear ineraction energy (LIE) approach
2008 G. Grazioso, Y.D. Pomè, C. Dallanoce, M. De Amici, C. De Micheli
Legenda icone
- file ad accesso aperto
- file disponibili sulla rete interna
- file disponibili agli utenti autorizzati
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile